SCHEMBL11244452

SCHEMBL11244452

CCCCCCCCc1ccc(N(c2ccc(CCCCCCCC)cc2)C2(c3ccc(N(C)C)cc3)OC(=O)c3ncccc32)cc1

nearest known ligand 0.36

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
TRPV1 Q8NER1 5/20 0.36
ALDH1A1 P00352 2/20 0.33
CYP3A4 P08684 2/20 0.33
HPGD P15428 2/20 0.33
CYP1A2 P05177 1/20 0.33
CYP2C19 P33261 1/20 0.33
KMT2A Q03164 1/20 0.33
CNR2 P34972 1/20 0.32
KAT2B Q92831 1/20 0.32
HIF1A Q16665 1/20 0.32
HSD17B10 Q99714 1/20 0.32
TDP1 Q9NUW8 1/20 0.32
THRA P10827 2/20 0.31
THRB P10828 2/20 0.31
SPHK1 Q9NYA1 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11249686 0.87 TRPV1 (0.34) TRPV1ALDH1A1CYP3A4HPGDCYP1A2
SCHEMBL11237226 0.84 TRPV1 (0.36) TRPV1ALDH1A1CYP3A4HPGDCYP1A2
SCHEMBL1882657 0.84 KMT2A (0.42) ALDH1A1CYP3A4HPGDCYP1A2CYP2C19
SCHEMBL11235932 0.83 ALDH1A1 (0.38) ALDH1A1CYP3A4HPGDCYP1A2CYP2C19
SCHEMBL11373082 0.81 ALDH1A1 (0.51) ALDH1A1CYP3A4HPGDCYP1A2CYP2C19
SCHEMBL11237151 0.81 LMNA (0.32) TRPV1CYP2C19CNR2
SCHEMBL11239963 0.78 CNR2 (0.36) TRPV1ALDH1A1CYP3A4HPGDCYP1A2
SCHEMBL11245349 0.77 GSK3A (0.36) ALDH1A1HPGDKMT2ACNR2KAT2B
SCHEMBL11228890 0.76 KMT2A (0.36) ALDH1A1HPGDCYP1A2CYP2C19KMT2A
SCHEMBL9462507 0.75 CYP2C19 (0.41) ALDH1A1CYP3A4HPGDCYP1A2CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4211872-A COLOR FORMERS FREEDOM CHEMICAL COMPANY 1980-07-08 US claimed
US-4337340-A FROM DIPHENYLAMINES AND BENZOYL OR 3-INDOLYLCARBONYL PYRIDINE- OR PYRAZINECARBOXYLIC ACIDS STERLING DRUG INC. (US) 1982-06-29 US disclosed
US-4243250-A FUROPYRIDINONES OR FUROPYRAZINONES AS COLOR FORMERS STERLING DRUG INC. (US) 1981-01-06 US disclosed
US-4211872-A COLOR FORMERS FREEDOM CHEMICAL COMPANY 1980-07-08 US disclosed