SCHEMBL11249066

SCHEMBL11249066

CCCCSC(=O)CCS(=O)(=O)CCCC

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
APEX1 P27695 1/20 0.37
NOS3 P29474 1/20 0.36
NOS1 P29475 1/20 0.36
NOS2 P35228 1/20 0.36
CES1 P23141 8/20 0.36
CES2 O00748 4/20 0.36
FAAH O00519 3/20 0.36
CA2 P00918 1/20 0.34
ALDH1A1 P00352 2/20 0.34
NPSR1 Q6W5P4 2/20 0.34
ESR1 P03372 1/20 0.33
ESR2 Q92731 1/20 0.33
LMNA P02545 2/20 0.32
NPC1 O15118 1/20 0.32
S1PR2 O95136 1/20 0.32
S1PR4 O95977 1/20 0.32
TP53 P04637 1/20 0.32
POLB P06746 1/20 0.32
MAPT P10636 1/20 0.32
HPGD P15428 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11475632 0.82 TDP1 (0.40) APEX1NOS3NOS1NOS2CES1
SCHEMBL11143545 0.79 NOS3 (0.48) NOS3NOS1NOS2CES1CES2
SCHEMBL3874809 0.77 NOS3 (0.46) NOS3NOS1NOS2CES1CES2
SCHEMBL26287322 0.77 CES1 (0.50) NOS3NOS1NOS2CES1CES2
SCHEMBL5127159 0.75 APEX1 (0.68) APEX1ALDH1A1NPSR1ESR1LMNA
SCHEMBL28288932 0.74 CES2 (0.52) CES1CES2ALDH1A1ESR1SMN1; SMN2
Acetone SCHEMBL9511697 0.74 CES1 (0.45) APEX1CES1CES2FAAHCA2
SCHEMBL7400053 0.74 FAAH (0.44) APEX1CES1CES2FAAHCA2
SCHEMBL52570 0.73 CA2 (0.52) CES1CES2FAAHCA2ALDH1A1
SCHEMBL11249064 0.73 CES1 (0.33) APEX1CES1CES2FAAHCA2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4323517-A ANTIPHLOGISTIC AGENTS TROPONWERKE GMBH & CO. KG (DE) 1982-04-06 US disclosed
US-4246278-A ANTIINFLAMMATORY SULFUR-CONTAINING ORGANIC ACIDS OR ESTERS OR THIOATES BAYER AKTIENGESELLSCHAFT (DE) 1981-01-20 US disclosed
EP-0002219-B1 MEDICINES WITH SULFUR CONTAINING ESTERS, AND THEIR PREPARATION Troponwerke GmbH & Co. KG (DE) 1980-12-10 EP disclosed
EP-0002219-A1 Medicines with sulfur containing esters, and their preparation Troponwerke GmbH & Co. KG (DE) 1979-06-13 EP disclosed