SCHEMBL11261678

SCHEMBL11261678

O=C(O)Cc1cccc2c(-c3ccc(Br)cc3)nccc12

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TDP1 Q9NUW8 1/20 0.45
ABCB11 O95342 1/20 0.42
LMNA P02545 1/20 0.42
PTGS1 P23219 1/20 0.42
ADORA1 P30542 1/20 0.42
PTGS2 P35354 1/20 0.42
KDM4E B2RXH2 3/20 0.42
MAPT P10636 2/20 0.42
ALDH1A1 P00352 2/20 0.42
ROS1 P08922 1/20 0.42
RPS6KB1 P23443 1/20 0.42
POLB P06746 1/20 0.42
CYP1A2 P05177 2/20 0.40
AKR1B1 P15121 3/20 0.38
CYP3A4 P08684 1/20 0.38
CYP2C9 P11712 1/20 0.38
CYP2C19 P33261 1/20 0.38
NPSR1 Q6W5P4 1/20 0.38
PTGDR2 Q9Y5Y4 5/20 0.38
AURKA O14965 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11500393 0.94 PTGDR2 (0.45) TDP1ABCB11LMNAPTGS1ADORA1
SCHEMBL11251835 0.89 TDP1 (0.54) TDP1KDM4EMAPTALDH1A1POLB
SCHEMBL11250127 0.87 IDO1 (0.47) TDP1LMNAKDM4EMAPTALDH1A1
SCHEMBL11246786 0.86 LMNA (0.48) TDP1LMNAKDM4EMAPTALDH1A1
SCHEMBL11255704 0.86 PTGDR2 (0.49) TDP1KDM4EMAPTALDH1A1POLB
SCHEMBL11262804 0.86 TDP1 (0.45) TDP1KDM4EMAPTPOLBCYP1A2
SCHEMBL11257966 0.85 ROS1 (0.46) KDM4EMAPTALDH1A1ROS1RPS6KB1
SCHEMBL11253776 0.85 ROS1 (0.41) TDP1LMNAKDM4EMAPTALDH1A1
SCHEMBL11249519 0.84 NPC1 (0.43) LMNAKDM4EMAPTALDH1A1ROS1
SCHEMBL11258880 0.83 MMP2 (0.51) TDP1PTGS1PTGS2KDM4EALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4337256-A ANTIINFLAMMATORY AGENTS; ANTIAGGLOMERANTS; ENZYME INHIBITORS; ANTIULCER AGENTS TEIKOKU HORMONE MANUFACTURING CO., LTD. (JP) 1982-06-29 US claimed
US-4337256-A ANTIINFLAMMATORY AGENTS; ANTIAGGLOMERANTS; ENZYME INHIBITORS; ANTIULCER AGENTS TEIKOKU HORMONE MANUFACTURING CO., LTD. (JP) 1982-06-29 US disclosed
EP-0013411-A1 Isoquinoline derivatives, process for their preparation and pharmaceutical compositions containing them TEIKOKU HORMONE MFG. CO., LTD. (JP) 1980-07-23 EP disclosed