SCHEMBL11266092

SCHEMBL11266092

CC(=O)OCc1cccc2c(-c3ccc(Br)cc3)nccc12

nearest known ligand 0.46

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
ROS1 P08922 1/20 0.37
RPS6KB1 P23443 1/20 0.37
L3MBTL1 Q9Y468 3/20 0.36
TRPV1 Q8NER1 2/20 0.36
TDP1 Q9NUW8 1/20 0.36
GPR84 Q9NQS5 2/20 0.35
ALDH1A1 P00352 2/20 0.34
MAOB P27338 2/20 0.34
MAOA P21397 1/20 0.34
MAPT P10636 1/20 0.34
GAA P10253 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11253776 0.81 ROS1 (0.41) ROS1RPS6KB1L3MBTL1TRPV1TDP1
SCHEMBL11249519 0.80 NPC1 (0.43) ROS1RPS6KB1L3MBTL1TRPV1GPR84
SCHEMBL11261678 0.80 TDP1 (0.45) ROS1RPS6KB1TRPV1TDP1ALDH1A1
SCHEMBL11257966 0.78 ROS1 (0.46) ROS1RPS6KB1L3MBTL1TRPV1ALDH1A1
SCHEMBL11258335 0.77 ALDH1A1 (0.39) ROS1RPS6KB1TRPV1GPR84ALDH1A1
SCHEMBL11256693 0.77 ALDH1A1 (0.39) ROS1RPS6KB1TRPV1GPR84ALDH1A1
SCHEMBL9685109 0.77 ALDH1A1 (0.53) L3MBTL1ALDH1A1MAPT
SCHEMBL11500393 0.75 PTGDR2 (0.45) ROS1RPS6KB1TDP1ALDH1A1MAPT
SCHEMBL11261674 0.73 TDO2 (0.36) ROS1RPS6KB1GPR84ALDH1A1
SCHEMBL11259590 0.72 TRPV1 (0.37) TRPV1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4337256-A ANTIINFLAMMATORY AGENTS; ANTIAGGLOMERANTS; ENZYME INHIBITORS; ANTIULCER AGENTS TEIKOKU HORMONE MANUFACTURING CO., LTD. (JP) 1982-06-29 US disclosed
EP-0013411-A1 Isoquinoline derivatives, process for their preparation and pharmaceutical compositions containing them TEIKOKU HORMONE MFG. CO., LTD. (JP) 1980-07-23 EP disclosed