SCHEMBL11257249

SCHEMBL11257249

O=C(NC(Cc1ccccc1)C(=O)N1CC1)OCc1ccccc1

nearest known ligand 0.63

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
TACR1 P25103 2/20 0.63
P2RX7 Q99572 11/20 0.61
CTSL P07711 1/20 0.58
CTSB P07858 1/20 0.58
CTSS P25774 1/20 0.58
CTSK P43235 1/20 0.58
ALDH1A1 P00352 1/20 0.57
ALOX15 P16050 1/20 0.57
TGM2 P21980 2/20 0.56

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11257246 1.00 TACR1 (0.63) TACR1P2RX7CTSLCTSBCTSS
SCHEMBL8750811 0.95 TACR1 (0.60) TACR1P2RX7CTSLCTSBCTSS
SCHEMBL8750802 0.95 TACR1 (0.60) TACR1P2RX7CTSLCTSBCTSS
SCHEMBL11232416 0.94 ITGB3 (0.62) TACR1P2RX7CTSLCTSBCTSS
SCHEMBL9483704 0.89 MC4R (0.61) TACR1P2RX7CTSLCTSBCTSS
SCHEMBL9483700 0.89 MC4R (0.61) TACR1P2RX7CTSLCTSBCTSS
SCHEMBL6349585 0.89 P2RX7 (0.73) P2RX7
SCHEMBL14305072 0.88 TGM2 (0.54) TACR1P2RX7CTSLCTSBCTSS
SCHEMBL6582593 0.87 CYP2C19 (0.62) TACR1P2RX7CTSLCTSBCTSS
SCHEMBL14790789 0.87 P2RX7 (0.53) TACR1P2RX7CTSLCTSBCTSK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0013790-B1 CLAVULANIC ACID DERIVATIVES, THEIR PREPARATION AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM BEECHAM GROUP PLC (GB) 1982-09-22 EP disclosed