SCHEMBL11258249

SCHEMBL11258249

CN1CCC(N2Cc3ccccc3Sc3ccccc32)CC1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP2D6 P10635 2/20 0.49
CYP1A2 P05177 1/20 0.49
KDM1A O60341 7/20 0.46
CHRM2 P08172 3/20 0.44
SIGMAR1 Q99720 2/20 0.44
CHRM3 P20309 2/20 0.44
ADRA2A P08913 2/20 0.44
CHRM1 P11229 2/20 0.44
DRD1 P21728 2/20 0.44
SLC6A2 P23975 2/20 0.44
SLC6A4 P31645 2/20 0.44
ADRA1A P35348 2/20 0.44
OPRM1 P35372 2/20 0.44
DRD3 P35462 2/20 0.44
SLC6A3 Q01959 2/20 0.44
KCNH2 Q12809 2/20 0.44
ABCB11 O95342 1/20 0.44
CHRM4 P08173 1/20 0.44
CHRM5 P08912 1/20 0.44
ADRA2B P18089 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11239038 0.86 PIM1 (0.46) CYP2D6CYP1A2KDM1ACHRM2SIGMAR1
SCHEMBL11098037 0.86 DRD2 (0.49) CYP2D6CYP1A2CHRM2SIGMAR1CHRM3
SCHEMBL11241659 0.86 CYP1A2 (0.42) CYP2D6CYP1A2KDM1ACHRM2SIGMAR1
SCHEMBL11247293 0.82 HTR2C (0.49) KDM1ASIGMAR1HTR2AHTR2CHTR2B
SCHEMBL9611568 0.80 CYP2D6 (0.55) CYP2D6CYP1A2KDM1ACHRM2SIGMAR1
SCHEMBL11103752 0.77 HTR2A (0.49) CYP2D6CYP1A2CHRM2CHRM3ADRA2A
SCHEMBL17933519 0.74 MAOA (0.55) CYP2D6CYP1A2KDM1ACHRM2SIGMAR1
SCHEMBL11256455 0.73 P2RX4 (0.48) CYP2D6CYP1A2CHRM2CHRM3OPRM1
SCHEMBL11633335 0.73 MAOA (0.50) CYP2D6CYP1A2KDM1ACHRM2SIGMAR1
SCHEMBL11246866 0.72 MAPT (0.56) CYP2D6CYP1A2KDM1ACHRM2SIGMAR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4360525-A NEUROLEPTIC AGENTS, ANTIDEPRESSANTS, SLEEP PROMOTERS SANDOZ LTD. (CH) 1982-11-23 US claimed