SCHEMBL11255746

SCHEMBL11255746

CNC(=O)Cc1cccc2c(C(C)C)nccc12

nearest known ligand 0.40

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.40
SMN1; SMN2 Q16637 2/20 0.40
LMNA P02545 3/20 0.38
ATM Q13315 1/20 0.38
ROS1 P08922 1/20 0.38
RPS6KB1 P23443 1/20 0.38
MEN1 O00255 2/20 0.37
KMT2A Q03164 2/20 0.37
CYP3A4 P08684 1/20 0.37
CYP2C19 P33261 1/20 0.37
RECQL P46063 1/20 0.37
MAPK10 P53779 5/20 0.37
MAPK8 P45983 4/20 0.37
MAPK9 P45984 4/20 0.37
KDM4E B2RXH2 1/20 0.37
GLS O94925 1/20 0.36
ACHE P22303 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11261355 0.84 TDP1 (0.50) ALDH1A1SMN1; SMN2KDM4E
SCHEMBL11257657 0.79 LMNA (0.46) SMN1; SMN2LMNAMEN1KMT2AKDM4E
SCHEMBL11254420 0.78 PKM (0.45) ALDH1A1SMN1; SMN2LMNAKMT2ARECQL
Formamide SCHEMBL11440222 0.78 TDP1 (0.44) ALDH1A1SMN1; SMN2CYP2C19KDM4E
SCHEMBL11267468 0.77 ANPEP (0.38) ALDH1A1MEN1KMT2ACYP3A4ACHE
SCHEMBL11257116 0.76 KMT2A (0.39) ALDH1A1LMNAATMMEN1KMT2A
SCHEMBL11257966 0.76 ROS1 (0.46) ALDH1A1SMN1; SMN2ATMROS1RPS6KB1
SCHEMBL11250074 0.74 LOXL2 (0.49) LMNAKDM4E
SCHEMBL11261342 0.74 GABRA1 (0.32) LMNAMEN1KMT2AKDM4E
SCHEMBL11249938 0.74 TDP1 (0.45) ALDH1A1SMN1; SMN2KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4337256-A ANTIINFLAMMATORY AGENTS; ANTIAGGLOMERANTS; ENZYME INHIBITORS; ANTIULCER AGENTS TEIKOKU HORMONE MANUFACTURING CO., LTD. (JP) 1982-06-29 US disclosed
EP-0013411-A1 Isoquinoline derivatives, process for their preparation and pharmaceutical compositions containing them TEIKOKU HORMONE MFG. CO., LTD. (JP) 1980-07-23 EP disclosed