SCHEMBL11263

SCHEMBL11263

COc1ccc(CNc2nc3ccc(B4OC(C)(C)C(C)(C)O4)cc3cc2CC(CC2CCCCC2)C(N)=O)cc1

nearest known ligand 0.36

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
HIF1A Q16665 2/20 0.36
NPC1 O15118 1/20 0.34
RAB9A P51151 1/20 0.34
SMN1; SMN2 Q16637 1/20 0.34
ALDH1A1 P00352 2/20 0.34
TDP1 Q9NUW8 2/20 0.34
TP53 P04637 1/20 0.34
MAPT P10636 1/20 0.34
CPB2 Q96IY4 1/20 0.34
KMT2A Q03164 1/20 0.34
SNCA P37840 1/20 0.33
BACE1 P56817 2/20 0.33
CTSS P25774 2/20 0.33
CTSL P07711 1/20 0.33
CTSK P43235 1/20 0.33
PDE10A Q9Y233 1/20 0.33
PPM1D O15297 1/20 0.32
VCP P55072 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8743 0.85 ALDH1A1 (0.38) NPC1RAB9ASMN1; SMN2ALDH1A1TDP1
SCHEMBL17620323 0.83 BACE1 (0.45) HIF1ANPC1RAB9ASMN1; SMN2ALDH1A1
SCHEMBL9169 0.80 BACE1 (0.45) TP53MAPTBACE1CTSSCTSL
SCHEMBL9716 0.79 BACE1 (0.37) ALDH1A1TDP1TP53CPB2KMT2A
SCHEMBL14702065 0.74 SNCA (0.45) HIF1ANPC1RAB9ASMN1; SMN2ALDH1A1
SCHEMBL14688444 0.73 PDE2A (0.45) RAB9AALDH1A1KMT2ASNCAPDE10A
SCHEMBL9498 0.71 KMT2A (0.42) NPC1RAB9ASMN1; SMN2ALDH1A1KMT2A
SCHEMBL14688581 0.70 RAB9A (0.45) NPC1RAB9ASMN1; SMN2ALDH1A1MAPT
SCHEMBL14688140 0.68 PDE1A (0.37) RAB9ATP53MAPTSNCA
SCHEMBL14688137 0.68 PDE1A (0.37) RAB9ATP53MAPTSNCA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2504315-A1 AMINO HETEROARYL COMPOUNDS AS BETA-SECRETASE MODULATORS AND METHODS OF USE Amgen Inc. (US) 2012-10-03 EP disclosed
WO-2011063233-A1 AMINO HETEROARYL COMPOUNDS AS BETA-SECRETASE MODULATORS AND METHODS OF USE AMGEN INC. (US) 2011-05-26 WO disclosed