SCHEMBL11265563

SCHEMBL11265563

CN(C)C(=N)NC(=O)Nc1ccc(O)c(O)c1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PYGL P06737 2/20 0.46
ALOX15 P16050 4/20 0.46
ERCC1 P07992 2/20 0.43
ERCC4 Q92889 2/20 0.43
SNCA P37840 1/20 0.42
TOP1 P11387 2/20 0.40
BCHE P06276 1/20 0.39
ACHE P22303 1/20 0.39
PIM1 P11309 1/20 0.39
ALDH1A1 P00352 2/20 0.38
APEX1 P27695 1/20 0.37
CYP1A2 P05177 2/20 0.37
CYP2D6 P10635 2/20 0.37
CYP2C9 P11712 2/20 0.37
CYP2C19 P33261 2/20 0.37
MEN1 O00255 1/20 0.37
CYP3A4 P08684 1/20 0.37
GAA P10253 1/20 0.37
KMT2A Q03164 1/20 0.37
PKM P14618 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14868432 0.84 SNCA (0.37) PYGLALOX15ERCC1ERCC4SNCA
SCHEMBL11269107 0.84 TOP1 (0.36) PYGLSNCATOP1ALDH1A1APEX1
SCHEMBL11280533 0.79 PYGL (0.47) PYGLALOX15ERCC1ERCC4SNCA
SCHEMBL11275768 0.79 PYGL (0.49) PYGLALOX15ERCC1ERCC4SNCA
SCHEMBL109020 0.77 ALOX15 (0.66) PYGLALOX15ERCC1ERCC4SNCA
SCHEMBL13804531 0.74 ALDH1A1 (0.55) PYGLALOX15ERCC1ERCC4SNCA
SCHEMBL10855224 0.74 MDM2 (0.58) BCHEALDH1A1MEN1KMT2APKM
SCHEMBL11276328 0.74 SNCA (0.41) ALOX15ERCC1ERCC4SNCATOP1
SCHEMBL11277145 0.72 SNCA (0.42) ALOX15ERCC1ERCC4SNCATOP1
SCHEMBL18155290 0.71 ALOX15 (0.55) PYGLALOX15ERCC1ERCC4SNCA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4326075-A ANTIDIARRHEA AGENTS WILLIAM H. RORER, INC. (US) 1982-04-20 US disclosed
US-4203920-A ANTIDIARRHEAL WILLIAM H. RORER, INC. (US) 1980-05-20 US disclosed
US-4060635-A Amidinoureas for treating diarrhea WILLIAM H. RORER, INC. (US) 1977-11-29 US disclosed