SCHEMBL11265587

SCHEMBL11265587

N#C/C=C/c1ccc(-c2ccccc2)cc1

nearest known ligand 0.52

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 2/20 0.52
CA1 P00915 1/20 0.48
MGLL Q99685 1/20 0.48
HDAC2 Q92769 2/20 0.44
HDAC1 Q13547 1/20 0.42
HDAC6 Q9UBN7 1/20 0.42
ENPP2 Q13822 1/20 0.42
TP53 P04637 1/20 0.39
ALDH1A1 P00352 1/20 0.39
ADORA1 P30542 1/20 0.39
FDPS P14324 1/20 0.38
NPC1 O15118 1/20 0.38
HPGD P15428 1/20 0.38
RAB9A P51151 1/20 0.38
SMN1; SMN2 Q16637 1/20 0.38
MAOB P27338 2/20 0.37
NFE2L2 Q16236 1/20 0.37
CYP19A1 P11511 1/20 0.37
MAOA P21397 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1287794 1.00 KDM4E (0.52) KDM4ECA1MGLLHDAC2HDAC1
Cinnamonitrile SCHEMBL28165460 0.91 ENPP2 (0.50) KDM4ECA1MGLLHDAC2HDAC1
SCHEMBL11125760 0.91 KDM4E (0.59) KDM4ECA1MGLLHDAC2HDAC1
SCHEMBL11304576 0.86 KDM4E (0.55) KDM4EHDAC1ENPP2MAOBNFE2L2
Cinnamonitrile SCHEMBL23599 0.86 KDM4E (0.54) KDM4ECA1HDAC2HDAC1HDAC6
Cinnamonitrile SCHEMBL996307 0.86 KDM4E (0.54) KDM4ECA1HDAC2HDAC1HDAC6
Cinnamonitrile SCHEMBL23933 0.86 KDM4E (0.54) KDM4ECA1HDAC2HDAC1HDAC6
SCHEMBL8904305 0.82 ENPP2 (0.54) KDM4EHDAC2HDAC1HDAC6ENPP2
SCHEMBL8904307 0.82 ENPP2 (0.54) KDM4EHDAC2HDAC1HDAC6ENPP2
SCHEMBL11293055 0.81 KDM4E (0.43) KDM4ECA1MGLLHDAC2HDAC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 18 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-111606824-B Beta-amino nitrile compound and preparation method thereof 东北师范大学 2023-03-14 CN claimed
CN-111606824-A Beta-amino nitrile compound and preparation method thereof 东北师范大学 2020-09-01 CN claimed
US-20230142654-A1 NOVEL COMPOUND, PREPARATION METHOD THEREOF, AND USE THEREOF PIMEDBIO, INC. (KR) 2023-05-11 US disclosed
US-20230142654-A1 NOVEL COMPOUND, PREPARATION METHOD THEREOF, AND USE THEREOF PIMEDBIO, INC. (KR) 2023-05-11 US disclosed
CN-111606824-B Beta-amino nitrile compound and preparation method thereof 东北师范大学 2023-03-14 CN disclosed
EP-3625218-B1 PROCESS FOR HYDROCYANATION OF TERMINAL ALKYNES STUDIENGESELLSCHAFT KOHLE MBH (DE) 2023-03-01 EP disclosed
EP-3625218-B1 PROCESS FOR HYDROCYANATION OF TERMINAL ALKYNES STUDIENGESELLSCHAFT KOHLE MBH (DE) 2023-03-01 EP disclosed
WO-2021145729-A1 NOVEL COMPOUND, PREPARATION METHOD THEREOF, AND USE THEREOF DAEGU-GYEONGBUK MEDICAL INNOVATION FOUNDATION (KR) 2021-07-22 WO disclosed
US-10947186-B2 Process for hydrocyanation of terminal alkynes STUDIENGESELLSCHAFT KOHLE MBH (DE) 2021-03-16 US disclosed
US-10947186-B2 Process for hydrocyanation of terminal alkynes STUDIENGESELLSCHAFT KOHLE MBH (DE) 2021-03-16 US disclosed
CN-111606824-A Beta-amino nitrile compound and preparation method thereof 东北师范大学 2020-09-01 CN disclosed
US-20200181068-A1 PROCESS FOR HYDROCYANATION OF TERMINAL ALKYNES STUDIENGESELLSCHAFT KOHLE MBH (DE) 2020-06-11 US disclosed
US-20200181068-A1 PROCESS FOR HYDROCYANATION OF TERMINAL ALKYNES STUDIENGESELLSCHAFT KOHLE MBH (DE) 2020-06-11 US disclosed
US-4336264-A 1-Benzoyl-3-(isoxazolyl or benzisoxazolyl)-ureas and insecticidal use thereof ELI LILLY AND COMPANY (US) 1982-06-22 US disclosed
US-4335054-A Process for the preparation of alkenylbenzenecarboxylic acid derivatives and alkenylnaphthalenecarboxylic acid derivatives CIBA-GEIGY CORPORATION (US) 1982-06-15 US disclosed
US-4322429-A Isoxazolylbenzamides as insecticides ELI LILLY AND COMPANY (US) 1982-03-30 US disclosed
EP-0048162-A1 Isoxazolylbenzamides ELI LILLY AND COMPANY (US) 1982-03-24 EP disclosed
EP-0042732-A1 1-benzoyl-3-substituted ureas and thioureas, their preparation, insecticidal formulations containing them and their use as insecticides ELI LILLY AND COMPANY (US) 1981-12-30 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20200181068-A1 PROCESS FOR HYDROCYANATION OF TERMINAL ALKYNES ALKBH3, ALKBH2, ALKBH5 KDM4E 154/4885CA1 3595/4885MGLL 1995/4885
US-20230142654-A1 NOVEL COMPOUND, PREPARATION METHOD THEREOF, AND USE THEREOF TYR, TYRO3, TH KDM4E 619/4885CA1 2779/4885MGLL 2997/4885
US-10947186-B2 Process for hydrocyanation of terminal alkynes ALKBH3, ALKBH2, ALKBH5 KDM4E 154/4885CA1 3595/4885MGLL 1995/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.