SCHEMBL11265804

SCHEMBL11265804

COc1ccc(N2CCN(CCCOc3ccc4c(c3)CCC4)CC2)cc1

nearest known ligand 0.68

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
ADRA1A P35348 3/20 0.68
ADRA1D P25100 2/20 0.68
ADRA1B P35368 2/20 0.68
MAPT P10636 2/20 0.65
TDP1 Q9NUW8 2/20 0.65
ALDH1A1 P00352 1/20 0.65
POLB P06746 1/20 0.65
HRH3 Q9Y5N1 7/20 0.63
HRH1 P35367 2/20 0.63
DRD2 P14416 5/20 0.60
HTR1A P08908 1/20 0.60
HTR2A P28223 1/20 0.60
HTR7 P34969 1/20 0.60
HSD17B10 Q99714 1/20 0.57
LMNA P02545 1/20 0.57
HTT P42858 1/20 0.57
DRD4 P21917 1/20 0.56
DRD3 P35462 1/20 0.56

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11268962 0.96 ADRA1A (0.67) ADRA1AADRA1DADRA1BMAPTTDP1
SCHEMBL11278148 0.90 KCNH2 (0.64) ADRA1AADRA1DADRA1BHRH3HRH1
SCHEMBL11274382 0.89 DRD2 (0.62) ADRA1AADRA1DADRA1BMAPTTDP1
SCHEMBL11271331 0.89 HRH3 (0.61) ADRA1AADRA1DADRA1BMAPTTDP1
SCHEMBL11269168 0.88 ADRA1D (0.68) ADRA1AADRA1DADRA1BHRH3HRH1
SCHEMBL11276891 0.88 HTR7 (0.66) ADRA1AADRA1DADRA1BHRH3HRH1
SCHEMBL11219235 0.88 HRH1 (0.80) ADRA1AMAPTTDP1HRH3HRH1
Hydrochloric Acid SCHEMBL11273968 0.87 HRH1 (0.78) ADRA1AMAPTTDP1HRH3HRH1
SCHEMBL11282931 0.86 HRH3 (0.67) HRH3HRH1
SCHEMBL11284279 0.85 HRH3 (0.59) ADRA1AADRA1DADRA1BMAPTTDP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4339580-A TRANQUILIZERS, SEDATIVES MITSUBISHI CHEMICAL INDUSTRIES, LIMITED (JP) 1982-07-13 US disclosed
EP-0021368-B1 PIPERAZINYLALKOXYINDANES AND ACID ADDITION SALTS THEREOF MITSUBISHI KASEI CORPORATION (JP) 1982-05-19 EP disclosed
EP-0021368-A1 Piperazinylalkoxyindanes and acid addition salts thereof MITSUBISHI KASEI CORPORATION (JP) 1981-01-07 EP disclosed