SCHEMBL11266451

SCHEMBL11266451

c1ccc(N2CCN(CCCCOc3ccc4c(c3)CCC4)CC2)cc1

nearest known ligand 0.74

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HRH1 P35367 3/20 0.74
HRH3 Q9Y5N1 1/20 0.74
DRD2 P14416 4/20 0.65
DRD3 P35462 3/20 0.64
HTR7 P34969 2/20 0.64
HTR1A P08908 3/20 0.61
HTR2A P28223 3/20 0.61
TMEM97 Q5BJF2 2/20 0.61
SIGMAR1 Q99720 2/20 0.61
SLC6A2 P23975 2/20 0.58
SLC6A4 P31645 2/20 0.58
MEN1 O00255 1/20 0.58
CYP1A2 P05177 1/20 0.58
CYP3A4 P08684 1/20 0.58
CYP2D6 P10635 1/20 0.58
MAPT P10636 1/20 0.58
CYP2C9 P11712 1/20 0.58
TSHR P16473 1/20 0.58
MAPK1 P28482 1/20 0.58
CYP2C19 P33261 1/20 0.58

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11219235 0.96 HRH1 (0.80) HRH1HRH3DRD2DRD3HTR7
Hydrochloric Acid SCHEMBL11273968 0.95 HRH1 (0.78) HRH1HRH3DRD2DRD3HTR7
SCHEMBL11285664 0.88 HTR7 (0.65) HRH1HRH3DRD2DRD3HTR7
SCHEMBL11277312 0.88 SLC6A2 (0.68) HRH1HRH3DRD2DRD3HTR1A
SCHEMBL11268962 0.88 ADRA1A (0.67) HRH1HRH3DRD2DRD3HTR7
SCHEMBL11278328 0.88 HRH1 (0.58) HRH1HRH3DRD2DRD3HTR7
SCHEMBL11278975 0.88 ADRA1D (0.68) HRH1HRH3DRD2HTR7SLC6A2
SCHEMBL6685654 0.85 HRH3 (1.00) HRH1HRH3DRD3KCNH2
SCHEMBL11278314 0.85 SLC6A4 (0.70) HRH1HRH3DRD2DRD3HTR7
SCHEMBL11285131 0.85 DRD2 (0.69) HRH1HRH3DRD2HTR7HTR2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4339580-A TRANQUILIZERS, SEDATIVES MITSUBISHI CHEMICAL INDUSTRIES, LIMITED (JP) 1982-07-13 US disclosed
EP-0021368-B1 PIPERAZINYLALKOXYINDANES AND ACID ADDITION SALTS THEREOF MITSUBISHI KASEI CORPORATION (JP) 1982-05-19 EP disclosed
EP-0021368-A1 Piperazinylalkoxyindanes and acid addition salts thereof MITSUBISHI KASEI CORPORATION (JP) 1981-01-07 EP disclosed