SCHEMBL11266780

SCHEMBL11266780

CC(=O)NC(=O)CSC(=O)c1cnc2ccccc2n1

nearest known ligand 0.50

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.48
HPGD P15428 1/20 0.48
ALOX15 P16050 1/20 0.48
HSD17B10 Q99714 1/20 0.48
KDM4E B2RXH2 2/20 0.47
HSP90AA1 P07900 1/20 0.47
HSP90AB1 P08238 1/20 0.47
SMN1; SMN2 Q16637 1/20 0.45
NPC1 O15118 2/20 0.43
RAB9A P51151 2/20 0.43
GRN P28799 1/20 0.43
SORT1 Q99523 1/20 0.43
GAA P10253 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11264480 0.75 KMT2A (0.60) ALDH1A1HPGDALOX15KDM4ESMN1; SMN2
SCHEMBL13928594 0.74 ALDH1A1 (0.62) ALDH1A1HPGDALOX15HSD17B10KDM4E
SCHEMBL11266631 0.73 SMN1; SMN2 (0.41) ALDH1A1HPGDHSD17B10SMN1; SMN2RAB9A
SCHEMBL11266339 0.72 KDM4E (0.41) ALDH1A1KDM4E
SCHEMBL4642665 0.71 ALDH1A1 (0.69) ALDH1A1HPGDALOX15HSD17B10KDM4E
SCHEMBL11267948 0.71 MAPT (0.51) ALDH1A1HPGDKDM4ESMN1; SMN2NPC1
SCHEMBL11266822 0.68 ALOX15 (0.53) ALDH1A1ALOX15HSD17B10SMN1; SMN2NPC1
SCHEMBL11267199 0.68 SMN1; SMN2 (0.44) ALDH1A1HPGDALOX15KDM4ESMN1; SMN2
SCHEMBL27347353 0.68 ALDH1A1 (0.74) ALDH1A1HPGDALOX15HSD17B10KDM4E
SCHEMBL12647223 0.67 ALDH1A1 (0.62) ALDH1A1HPGDALOX15HSD17B10SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4329363-A Substituted mercapto acid amides and their use MERCK & CO., INC. (US) 1982-05-11 US disclosed
US-4216160-A IMMUNOREGULANTS FOR CORRECTING AN INBALANCE OF IMMUNE HOMEOSTASIS MERCK & CO., INC. (US) 1980-08-05 US disclosed