SCHEMBL11270104

SCHEMBL11270104

Clc1cc2c(cc1OCCCN1CCN(c3ccccc3)CC1)CCC2

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR1A P08908 7/20 0.56
DRD3 P35462 5/20 0.56
DRD2 P14416 4/20 0.56
HTR2A P28223 4/20 0.56
TMEM97 Q5BJF2 3/20 0.56
SIGMAR1 Q99720 3/20 0.56
HRH1 P35367 3/20 0.56
HTR7 P34969 1/20 0.56
ADRA1A P35348 1/20 0.56
HRH3 Q9Y5N1 2/20 0.55
KCNH2 Q12809 1/20 0.50
HTR4 Q13639 1/20 0.49
MEN1 O00255 1/20 0.48
CYP1A2 P05177 1/20 0.48
CYP3A4 P08684 1/20 0.48
CYP2D6 P10635 1/20 0.48
MAPT P10636 1/20 0.48
CYP2C9 P11712 1/20 0.48
TSHR P16473 1/20 0.48
MAPK1 P28482 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11275227 0.90 KCNH2 (0.60) DRD3DRD2SIGMAR1HTR7ADRA1A
SCHEMBL11274363 0.88 DRD2 (0.59) HTR1ADRD3DRD2HTR2ATMEM97
SCHEMBL11300075 0.86 KCNH2 (0.62) HTR1ADRD2HTR2ASIGMAR1HTR7
SCHEMBL11266553 0.86 HTR1A (0.62) HTR1ADRD3DRD2HTR2ATMEM97
SCHEMBL11292019 0.86 TSHR (0.59) HTR1ADRD3DRD2HTR2ATMEM97
SCHEMBL11270622 0.86 DRD3 (0.57) HTR1ADRD3DRD2HTR2ATMEM97
SCHEMBL11280762 0.86 DRD3 (0.56) HTR1ADRD3DRD2HTR2ATMEM97
SCHEMBL11273088 0.85 SLC6A4 (0.52) HTR1ADRD3DRD2HTR2ATMEM97
Hydrochloric Acid SCHEMBL11284442 0.85 HTR1A (0.56) HTR1ADRD3DRD2HTR2ATMEM97
SCHEMBL11297779 0.85 DRD2 (0.55) HTR1ADRD3DRD2HTR2AADRA1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4339580-A TRANQUILIZERS, SEDATIVES MITSUBISHI CHEMICAL INDUSTRIES, LIMITED (JP) 1982-07-13 US disclosed
EP-0021368-B1 PIPERAZINYLALKOXYINDANES AND ACID ADDITION SALTS THEREOF MITSUBISHI KASEI CORPORATION (JP) 1982-05-19 EP disclosed
EP-0021368-A1 Piperazinylalkoxyindanes and acid addition salts thereof MITSUBISHI KASEI CORPORATION (JP) 1981-01-07 EP disclosed