SCHEMBL11280762

SCHEMBL11280762

COc1cc2c(cc1OCCCN1CCN(c3ccccc3)CC1)CCC2

nearest known ligand 0.56

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
DRD3 P35462 4/20 0.56
HTR1A P08908 4/20 0.56
HRH1 P35367 3/20 0.56
DRD2 P14416 2/20 0.56
HTR2A P28223 2/20 0.56
TMEM97 Q5BJF2 2/20 0.56
SIGMAR1 Q99720 2/20 0.56
HRH3 Q9Y5N1 2/20 0.55
BCHE P06276 1/20 0.52
ACHE P22303 1/20 0.52
HTR4 Q13639 1/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11266112 0.88 ABCB1 (0.55) DRD3HTR1AHRH1DRD2HTR2A
SCHEMBL11266553 0.88 HTR1A (0.62) DRD3HTR1AHRH1DRD2HTR2A
SCHEMBL11283459 0.88 KCNH2 (0.60) SIGMAR1
SCHEMBL11292019 0.86 TSHR (0.59) DRD3HTR1AHRH1DRD2HTR2A
SCHEMBL11270622 0.86 DRD3 (0.57) DRD3HTR1AHRH1DRD2HTR2A
SCHEMBL11270104 0.86 HTR1A (0.56) DRD3HTR1AHRH1DRD2HTR2A
SCHEMBL11271731 0.85 SLC6A4 (0.52) DRD3HTR1ADRD2HTR2ASIGMAR1
SCHEMBL11282244 0.85 DRD2 (0.53) DRD3HTR1AHRH1DRD2HTR2A
SCHEMBL11273685 0.85 HTR2A (0.53) DRD3HTR1ADRD2HTR2AHTR4
Hydrochloric Acid SCHEMBL11284442 0.85 HTR1A (0.56) DRD3HTR1AHRH1DRD2HTR2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4339580-A TRANQUILIZERS, SEDATIVES MITSUBISHI CHEMICAL INDUSTRIES, LIMITED (JP) 1982-07-13 US disclosed
EP-0021368-B1 PIPERAZINYLALKOXYINDANES AND ACID ADDITION SALTS THEREOF MITSUBISHI KASEI CORPORATION (JP) 1982-05-19 EP disclosed
EP-0021368-A1 Piperazinylalkoxyindanes and acid addition salts thereof MITSUBISHI KASEI CORPORATION (JP) 1981-01-07 EP disclosed