SCHEMBL11270280

SCHEMBL11270280

Cc1cc(F)ccc1NC(=O)NC(=N)N

nearest known ligand 0.48

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
CHIT1 Q13231 1/20 0.48
HTT P42858 4/20 0.48
ALDH1A1 P00352 3/20 0.48
MAPT P10636 3/20 0.48
LMNA P02545 2/20 0.48
SMN1; SMN2 Q16637 2/20 0.48
MEN1 O00255 1/20 0.48
KMT2A Q03164 1/20 0.48
NPSR1 Q6W5P4 1/20 0.48
POLB P06746 1/20 0.46
KDM4E B2RXH2 2/20 0.45
SIGMAR1 Q99720 1/20 0.44
RAB9A P51151 3/20 0.43
NPC1 O15118 2/20 0.43
TRPV1 Q8NER1 1/20 0.42
PKM P14618 1/20 0.40
PYGL P06737 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11412037 0.84 SIGMAR1 (0.46) CHIT1HTTALDH1A1MAPTLMNA
SCHEMBL11320624 0.84 RAB9A (0.56) HTTALDH1A1MAPTLMNASMN1; SMN2
SCHEMBL11052921 0.84 MEN1 (0.56) HTTALDH1A1MAPTLMNASMN1; SMN2
SCHEMBL11882906 0.84 SIGMAR1 (0.50) CHIT1HTTALDH1A1MAPTLMNA
SCHEMBL11285564 0.82 PKM (0.53) HTTALDH1A1MAPTSMN1; SMN2MEN1
Methylamine SCHEMBL11259444 0.82 SIGMAR1 (0.49) CHIT1HTTALDH1A1MAPTLMNA
SCHEMBL11320603 0.82 CA1 (0.44) HTTALDH1A1MAPTSMN1; SMN2MEN1
SCHEMBL11254202 0.82 ALDH1A1 (0.46) CHIT1HTTALDH1A1MAPTLMNA
SCHEMBL11140703 0.82 NOX1 (0.47) CHIT1HTTALDH1A1MAPTSMN1; SMN2
SCHEMBL11313322 0.82 PYGL (0.55) KMT2ANPSR1PYGL

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4326075-A ANTIDIARRHEA AGENTS WILLIAM H. RORER, INC. (US) 1982-04-20 US disclosed
US-4216229-A 1-AMIDINO-3-PHENYLUREAS WILLIAM H. RORER, INC. (US) 1980-08-05 US disclosed
US-4216230-A Method for alleviating hypertension with amidinoureas WILLIAM H. RORER, INC. (US) 1980-08-05 US disclosed
US-4203920-A ANTIDIARRHEAL WILLIAM H. RORER, INC. (US) 1980-05-20 US disclosed
US-4150154-A GASTROINTESTINAL ANTISPASMODICS WILLIAM H. RORER, INC. (US) 1979-04-17 US disclosed
US-4060635-A Amidinoureas for treating diarrhea WILLIAM H. RORER, INC. (US) 1977-11-29 US disclosed