SCHEMBL11273008

SCHEMBL11273008

c1ccc(Oc2nnc(-c3ccccc3)c(-c3ccccc3)n2)cc1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADORA2A P29274 5/20 0.50
ADORA1 P30542 4/20 0.50
ALDH1A1 P00352 7/20 0.46
LMNA P02545 4/20 0.46
NPSR1 Q6W5P4 4/20 0.46
SMN1; SMN2 Q16637 3/20 0.46
KDM4E B2RXH2 2/20 0.46
GAA P10253 1/20 0.46
MAPT P10636 3/20 0.43
MEN1 O00255 4/20 0.42
KMT2A Q03164 4/20 0.42
HTT P42858 1/20 0.41
GPR55 Q9Y2T6 1/20 0.41
GLA P06280 1/20 0.41
POLB P06746 1/20 0.41
HPGD P15428 1/20 0.41
LTA4H P09960 1/20 0.41
TSHR P16473 1/20 0.41
TDP1 Q9NUW8 1/20 0.41
L3MBTL1 Q9Y468 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11337491 0.88 ALDH1A1 (0.57) ADORA2AADORA1ALDH1A1LMNANPSR1
SCHEMBL28303870 0.78 ADORA2A (0.52) ADORA2AADORA1ALDH1A1LMNANPSR1
SCHEMBL11268851 0.78 SMN1; SMN2 (0.53) ADORA2AADORA1ALDH1A1LMNANPSR1
SCHEMBL11273639 0.74 GPR84 (0.49) ADORA2AADORA1ALDH1A1LMNANPSR1
SCHEMBL11280072 0.74 NPSR1 (0.47) ADORA2AADORA1ALDH1A1LMNANPSR1
SCHEMBL1006428 0.71 PAX8 (0.63) ALDH1A1SMN1; SMN2KDM4EGAAMAPT
SCHEMBL24124452 0.71 SMN1; SMN2 (0.54) ALDH1A1LMNASMN1; SMN2KDM4EGAA
SCHEMBL22724736 0.71 SMN1; SMN2 (0.54) ALDH1A1LMNASMN1; SMN2KDM4EGAA
SCHEMBL14280962 0.71 ADORA2A (0.54) ADORA2AALDH1A1LMNANPSR1SMN1; SMN2
SCHEMBL11778554 0.69 MAPK1 (0.56) ADORA2AADORA1ALDH1A1NPSR1SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4310551-A Pharmacologically active substituted 1,2,4-triazines DIAMOND SHAMROCK CORPORATION (US) 1982-01-12 US disclosed
US-4251527-A ANTIINFLAMMATORY AGENTS DIAMOND SHAMROCK CORPORATION (US) 1981-02-17 US disclosed
US-4157392-A HYPOTENSIVE AGENTS, ANTIINFLAMMATORY AGENTS, ANALGESICS, ANTIPYRETICS AND NERVOUS SYSTEM EFFECTS DIAMOND SHAMROCK CORPORATION (US) 1979-06-05 US disclosed