SCHEMBL1128920

SCHEMBL1128920

CC(C)c1cccc2[nH]c(Cl)nc12

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 1/20 0.46
RAB9A P51151 1/20 0.46
LMNA P02545 2/20 0.45
EGFR P00533 1/20 0.38
MGAM O43451 3/20 0.37
GAA P10253 3/20 0.37
SI P14410 3/20 0.37
MGAM2 Q2M2H8 3/20 0.37
PSMB8 P28062 1/20 0.37
GABRA1 P14867 2/20 0.36
GABRG2 P18507 2/20 0.36
GABRB3 P28472 2/20 0.36
FAAH O00519 1/20 0.36
CA1 P00915 1/20 0.36
CA2 P00918 1/20 0.36
CYP1A2 P05177 1/20 0.36
CYP3A4 P08684 1/20 0.36
HPGD P15428 1/20 0.36
TSHR P16473 1/20 0.36
GABRB1 P18505 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7246922 0.81 NPC1 (0.40) NPC1RAB9AMGAMGAASI
SCHEMBL7261494 0.81 CXCL8 (0.43) NPC1RAB9AHPGDPTGS1PARP1
SCHEMBL24995382 0.80 HSD17B10 (0.49) LMNAEGFRGABRA1GABRG2GABRB3
SCHEMBL13192695 0.80 PARP1 (0.50) LMNAEGFRMGAMGAASI
SCHEMBL15111522 0.80 PARP1 (0.44) NPC1RAB9APARP1
SCHEMBL20315207 0.79 NUDT1 (0.47) LMNAEGFRGAAGABRA1GABRG2
SCHEMBL9305449 0.79 LMNA (0.38) LMNAEGFRMGAMGAASI
SCHEMBL19002278 0.79 GABRA1 (0.45) LMNAEGFRMGAMGAASI
SCHEMBL8713612 0.79 LMNA (0.38) LMNAEGFRMGAMGAASI
SCHEMBL10694372 0.78 LMNA (0.45) LMNAEGFRGABRA1GABRG2GABRB3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2282762-A2 NOVEL MACROCYCLIC INHIBITORS OF HEPATITIS C VIRUS REPLICATION Intermune, Inc. (US) 2011-02-16 EP disclosed
WO-2009142842-A2 NOVEL MACROCYCLIC INHIBITORS OF HEPATITIS C VIRUS REPLICATION INTERMUNE, INC. (US) 2009-11-26 WO disclosed
EP-0039190-A1 2-(1-Piperazinyl)-4-pyrimidinamines and related compounds AMERICAN HOME PRODUCTS CORPORATION (US) 1981-11-04 EP disclosed