SCHEMBL1129405

SCHEMBL1129405

O=C[C@@H](OC(=O)O)[C@H](O)[C@H](O)CO

nearest known ligand 0.42

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
PDE4A P27815 1/20 0.42
LMNA P02545 2/20 0.39
USP2 O75604 1/20 0.39
SLCO1B1 Q9Y6L6 1/20 0.39
L3MBTL1 Q9Y468 1/20 0.39
TDP1 Q9NUW8 1/20 0.37
AKR1B1 P15121 1/20 0.34
OR51E2 Q9H255 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1607591 1.00 PDE4A (0.42) PDE4ALMNAUSP2SLCO1B1L3MBTL1
SCHEMBL2122285 0.98 PDE4A (0.41) PDE4ALMNAUSP2SLCO1B1L3MBTL1
SCHEMBL419462 0.94 PDE4A (0.45) PDE4ALMNAUSP2SLCO1B1L3MBTL1
SCHEMBL10738624 0.94 PDE4A (0.45) PDE4ALMNAUSP2SLCO1B1L3MBTL1
SCHEMBL17144674 0.94 PDE4A (0.45) PDE4ALMNAUSP2SLCO1B1L3MBTL1
SCHEMBL18730385 0.92 PDE4A (0.44) PDE4ALMNAUSP2SLCO1B1L3MBTL1
SCHEMBL1537561 0.92 PDE4A (0.44) PDE4ALMNAUSP2SLCO1B1L3MBTL1
SCHEMBL10743488 0.92 TDP1 (0.44) PDE4ALMNAUSP2SLCO1B1L3MBTL1
SCHEMBL8384985 0.87 PDE4A (0.38) PDE4ALMNAUSP2SLCO1B1L3MBTL1
SCHEMBL1257816 0.84 LMNA (0.39) PDE4ALMNAUSP2SLCO1B1L3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 17 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2282773-B2 METHODS AND COMPOSITIONS FOR MAKING ANTIBODIES AND ANTIBODY DERIVATIVES WITH REDUCED CORE FUCOSYLATION SEAGEN INC (US) 2025-03-05 EP disclosed
US-20230055475-A1 METHODS AND COMPOSITIONS FOR MAKING ANTIBODIES AND ANTIBODY DERIVATIVES WITH REDUCED CORE FUCOSYLATION SEAGEN INC (US) 2023-02-23 US disclosed
US-11319526-B2 Methods and compositions for making antibodies and antibody derivatives with reduced core fucosylation SEAGEN INC. (US) 2022-05-03 US disclosed
US-10443035-B2 Methods and compositions for making antibodies and antibody derivatives with reduced core fucosylation SEATTLE GENETICS, INC. (US) 2019-10-15 US disclosed
US-20190276796-A1 METHODS AND COMPOSITIONS FOR MAKING ANTIBODIES AND ANTIBODY DERIVATIVES WITH REDUCED CORE FUCOSYLATION SEAGEN INC. 2019-09-12 US disclosed
US-20180155677-A1 METHODS AND COMPOSITIONS FOR MAKING ANTIBODIES AND ANTIBODY DERIVATIVES WITH REDUCED CORE FUCOSYLATION SEAGEN INC. 2018-06-07 US disclosed
US-9816069-B2 Methods and compositions for making antibodies and antibody derivatives with reduced core fucosylation SEATTLE GENETICS, INC. (US) 2017-11-14 US disclosed
US-20150337259-A1 METHODS AND COMPOSITIONS FOR MAKING ANTIBODIES AND ANTIBODY DERIVATIVES WITH REDUCED CORE FUCOSYLATION SEAGEN INC. 2015-11-26 US disclosed
US-8993326-B2 Methods and compositions for making antibodies and antibody derivatives with reduced core fucosylation SEATTLE GENETICS, INC. (US) 2015-03-31 US disclosed
US-20140031536-A1 METHODS AND COMPOSITIONS FOR MAKING ANTIBODIES AND ANTIBODY DERIVATIVES WITH REDUCED CORE FUCOSYLATION SEATTLE GENETICS, INC. (US) 2014-01-30 US disclosed
EP-2282773-B1 METHODS AND COMPOSITIONS FOR MAKING ANTIBODIES AND ANTIBODY DERIVATIVES WITH REDUCED CORE FUCOSYLATION SEATTLE GENETICS INC (US) 2014-01-15 EP disclosed
US-8574907-B2 Methods and compositions for making antibodies and antibody derivatives with reduced core fucosylation SEATTLE GENETICS, INC. (US) 2013-11-05 US disclosed
US-20120183997-A1 METHODS AND COMPOSITIONS FOR MAKING ANTIBODIES AND ANTIBODY DERIVATIVES WITH REDUCED CORE FUCOSYLATION SEATTLE GENETICS, INC. (US) 2012-07-19 US disclosed
US-8163551-B2 Methods and compositions for making antibodies and antibody derivatives with reduced core fucosylation SEATTLE GENETICS, INC. (US) 2012-04-24 US disclosed
EP-2282773-A2 METHODS AND COMPOSITIONS FOR MAKING ANTIBODIES AND ANTIBODY DERIVATIVES WITH REDUCED CORE FUCOSYLATION Seattle Genetics, Inc. (US) 2011-02-16 EP disclosed
US-20090317869-A1 METHODS AND COMPOSITIONS FOR MAKING ANTIBODIES AND ANTIBODY DERIVATIVES WITH REDUCED CORE FUCOSYLATION SEATTLE GENETICS, INC. (US) 2009-12-24 US disclosed
WO-2009135181-A2 METHODS AND COMPOSITIONS FOR MAKING ANTIBODIES AND ANTIBODY DERIVATIVES WITH REDUCED CORE FUCOSYLATION SEATTLE GENETICS, INC. (US) 2009-11-05 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (6 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20140031536-A1 METHODS AND COMPOSITIONS FOR MAKING ANTIBODIES AND ANTIBODY DERIVATIVES WITH REDUCED CORE FUCOSYLATION FUT5, FUCA2, FCGR3B PDE4A 4544/4885LMNA 2329/4885USP2 1994/4885
US-20180155677-A1 METHODS AND COMPOSITIONS FOR MAKING ANTIBODIES AND ANTIBODY DERIVATIVES WITH REDUCED CORE FUCOSYLATION FUT5, FUCA2, FCGR3B PDE4A 4544/4885LMNA 2329/4885USP2 1994/4885
US-20230055475-A1 METHODS AND COMPOSITIONS FOR MAKING ANTIBODIES AND ANTIBODY DERIVATIVES WITH REDUCED CORE FUCOSYLATION FUT5, FUCA2, FCGR3B PDE4A 4544/4885LMNA 2329/4885USP2 1994/4885
US-10443035-B2 Methods and compositions for making antibodies and antibody derivatives with reduced core fucosylation FUT5, FUCA2, FCGR3B PDE4A 4544/4885LMNA 2329/4885USP2 1994/4885
US-20190276796-A1 METHODS AND COMPOSITIONS FOR MAKING ANTIBODIES AND ANTIBODY DERIVATIVES WITH REDUCED CORE FUCOSYLATION FUT5, FUCA2, FCGR3B PDE4A 4544/4885LMNA 2329/4885USP2 1994/4885
US-11319526-B2 Methods and compositions for making antibodies and antibody derivatives with reduced core fucosylation FUT5, FUCA2, FCGR3B PDE4A 4544/4885LMNA 2329/4885USP2 1994/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.