SCHEMBL11296003

SCHEMBL11296003

O=C(O)c1ccc(-c2ccccc2)cc1CBr

nearest known ligand 0.70

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DCLRE1B Q9H816 3/20 0.70
DCLRE1A Q6PJP8 1/20 0.70
ACMSD Q8TDX5 3/20 0.58
HNF4A P41235 2/20 0.58
ACLY P53396 4/20 0.53
DHFR P00374 1/20 0.53
MCL1 Q07820 1/20 0.53
PTPN1 P18031 4/20 0.51
PTPN2 P17706 1/20 0.51
PTPN6 P29350 1/20 0.51
KMO O15229 1/20 0.47
GSK3B P49841 1/20 0.46
GRIN2D O15399 1/20 0.45
GRIN2A Q12879 1/20 0.45
GRIN2B Q13224 1/20 0.45
GRIN2C Q14957 1/20 0.45
AKR1C4 P17516 1/20 0.45
AKR1C3 P42330 1/20 0.45
AKR1C2 P52895 1/20 0.45
AKR1C1 Q04828 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10397478 0.84 DCLRE1B (0.72) DCLRE1BDCLRE1AACMSDHNF4AACLY
SCHEMBL14084578 0.82 NR4A2 (0.51) DCLRE1BDCLRE1AACMSDHNF4AACLY
Hydrochloric Acid SCHEMBL5704000 0.80 DCLRE1B (0.62) DCLRE1BDCLRE1AACMSDHNF4AACLY
SCHEMBL12991938 0.80 TSHR (0.51) DCLRE1BDCLRE1A
SCHEMBL7019419 0.79 DCLRE1B (0.66) DCLRE1BDCLRE1AACMSDHNF4AACLY
SCHEMBL13681701 0.79 DCLRE1B (0.66) DCLRE1BDCLRE1AACMSDHNF4AACLY
SCHEMBL28180523 0.77 KDM4E (0.48) DCLRE1BDCLRE1APTPN1
SCHEMBL26679439 0.77 DCLRE1B (0.62) DCLRE1BDCLRE1AACMSDHNF4AACLY
SCHEMBL445508 0.77 FOLH1 (0.59) AKR1C3
SCHEMBL30616786 0.77 ACMSD (0.70) DCLRE1BDCLRE1AACMSDHNF4AACLY

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2665744-A2 MACROCYCLIC COMPOUNDS WITH A HYBRID PEPTIDIC/NON-PEPTIDIC BACKBONE AND METHODS FOR THEIR PREPARATION UNIVERSITY OF ROCHESTER (US) 2013-11-27 EP disclosed
WO-2012100176-A2 MACROCYCLIC COMPOUNDS WITH A HYBRID PEPTIDIC/NON-PEPTIDIC BACKBONE AND METHODS FOR THEIR PREPARATION UNIVERSITY OF ROCHESTER (US) 2012-07-26 WO disclosed