SCHEMBL11297451

SCHEMBL11297451

C=CC(=O)CC(c1ccc(SC)cc1)N1CCOCC1

nearest known ligand 0.51

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.46
TSHR P16473 2/20 0.46
HTT P42858 1/20 0.46
MAPK1 P28482 1/20 0.42
SMN1; SMN2 Q16637 1/20 0.42
THRB P10828 2/20 0.39
P2RX7 Q99572 6/20 0.38
TP53 P04637 3/20 0.38
MAPT P10636 3/20 0.37
LMNA P02545 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL11294182 0.99 ALDH1A1 (0.45) ALDH1A1TSHRHTTMAPK1SMN1; SMN2
SCHEMBL11293575 0.85 ALDH1A1 (0.46) ALDH1A1TSHRSMN1; SMN2THRBP2RX7
SCHEMBL3051654 0.84 P2RX7 (0.50) THRBP2RX7TP53MAPTLMNA
Hydrochloric Acid SCHEMBL11299080 0.84 ALDH1A1 (0.45) ALDH1A1TSHRSMN1; SMN2THRBP2RX7
SCHEMBL3051670 0.81 P2RX7 (0.48) ALDH1A1HTTSMN1; SMN2THRBP2RX7
SCHEMBL22660960 0.78 ALDH1A1 (0.45) ALDH1A1TSHRHTTMAPK1SMN1; SMN2
SCHEMBL3047241 0.78 SLC6A2 (0.55) ALDH1A1SMN1; SMN2P2RX7
SCHEMBL28210928 0.77 ALDH1A1 (0.45) ALDH1A1TSHRHTTMAPK1SMN1; SMN2
SCHEMBL3040850 0.72 DPP4 (0.46) P2RX7LMNA
SCHEMBL3260671 0.72 LMNA (0.44) ALDH1A1LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0043141-A1 Pharmaceutical compositions having antiviral activity for topical administration and the use of 1-(substituted phenyl)-5-(4-morpholinyl)-1-penten-3-one compounds for the preparation of pharmaceutical compositions having an antiviral effect MERRELL DOW PHARMACEUTICALS INC. (US) 1982-01-06 EP disclosed