SCHEMBL11337486

SCHEMBL11337486

O=C(Nc1ccc(C(=O)Nc2c(O)c(S(=O)(=O)O)cc3ccccc23)cc1)Nc1ccc(C(=O)Nc2c(O)c(S(=O)(=O)O)cc3ccccc23)cc1

nearest known ligand 0.48

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
TIMP3 P35625 2/20 0.47
FGF1 P05230 1/20 0.47
PRMT1 Q99873 2/20 0.47
PRMT3 O60678 1/20 0.47
EP300 Q09472 1/20 0.47
PRMT6 Q96LA8 1/20 0.47
SIRT1 Q96EB6 2/20 0.44
ENPP2 Q13822 3/20 0.43
POLB P06746 1/20 0.42
DEGS1 O15121 1/20 0.42
CD40 P25942 2/20 0.42
CD40LG P29965 2/20 0.42
RAB9A P51151 1/20 0.41
KMT2A Q03164 1/20 0.41
FLT3 P36888 2/20 0.41
HPSE Q9Y251 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10908400 0.93 DEGS1 (0.42) TIMP3FGF1PRMT1PRMT3EP300
SCHEMBL11338609 0.90 PRMT1 (0.49) TIMP3FGF1PRMT1PRMT3EP300
SCHEMBL11350543 0.88 KMT2A (0.52) TIMP3PRMT1SIRT1POLBRAB9A
SCHEMBL11427755 0.86 CASP6 (0.48) PRMT1POLBRAB9AKMT2A
SCHEMBL10907652 0.83 PRMT1 (0.42) TIMP3FGF1PRMT1PRMT3EP300
SCHEMBL11341867 0.83 DHODH (0.44) TIMP3PRMT1SIRT1POLBRAB9A
SCHEMBL11344837 0.83 PRMT1 (0.43) PRMT1PRMT3EP300PRMT6ENPP2
SCHEMBL11347286 0.82 TIMP3 (0.49) TIMP3FGF1PRMT1PRMT3EP300
SCHEMBL11437915 0.82 CD40 (0.54) PRMT1POLBCD40CD40LGRAB9A
SCHEMBL10823709 0.82 LMNA (0.52) PRMT1PRMT3EP300PRMT6ENPP2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4297372-A ANTIARTHRITIC AGENTS; COLLAGENASE AND PROTEOLYTIC ENZYME INHIBITORS; BONE, SKIN, AND ORAL DISORDERS AMERICAN CYANAMID COMPANY (US) 1981-10-27 US disclosed
EP-0013784-A1 C-Substituted naphthalenemonosulfonic ureides, process for their preparation and pharmaceutical compositions containing them AMERICAN CYANAMID COMPANY (US) 1980-08-06 EP disclosed
US-4216164-A Ureide inhibitors of connective tissue destruction AMERICAN CYANAMID COMPANY (US) 1980-08-05 US disclosed