SCHEMBL11344993

SCHEMBL11344993

O=C(C1=CCCN1)c1cccs1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DAO P14920 1/20 0.48
HPGDS O60760 1/20 0.47
CES2 O00748 1/20 0.46
CES1 P23141 1/20 0.46
HPGD P15428 5/20 0.44
LMNA P02545 3/20 0.44
HTT P42858 2/20 0.44
ALOX15 P16050 2/20 0.44
ALDH1A1 P00352 5/20 0.42
NPC1 O15118 5/20 0.42
RAB9A P51151 5/20 0.42
MEN1 O00255 4/20 0.42
KMT2A Q03164 4/20 0.42
POLB P06746 2/20 0.42
HDAC1 Q13547 1/20 0.42
TP53 P04637 3/20 0.41
SMN1; SMN2 Q16637 3/20 0.41
GAA P10253 2/20 0.41
HSD17B10 Q99714 2/20 0.41
NFKB1 P19838 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28324811 0.79 HPGDS (0.46) DAOHPGDSCES2CES1HPGD
SCHEMBL182010 0.73 CES2 (0.71) DAOHPGDSCES2CES1HPGD
Cyclopentane SCHEMBL8081415 0.72 HPGDS (0.63) DAOHPGDSCES2CES1HPGD
Thiophene Carboxylic Acid SCHEMBL28789119 0.69 DAO (0.76) DAOHPGDSCES2CES1HPGD
Piperazine SCHEMBL28327330 0.68 ALDH1A1 (0.45) DAOCES2CES1ALDH1A1RAB9A
SCHEMBL6793430 0.68 HPGDS (0.83) DAOHPGDSCES2CES1HPGD
Thiophene Carboxylic Acid SCHEMBL7062244 0.67 DAO (1.00) DAOHPGDSCES2CES1HPGD
SCHEMBL225933 0.67
Thiophene Carboxylic Acid SCHEMBL83000 0.67
Thiophene Carboxylic Acid SCHEMBL27774764 0.67 DAO (1.00) DAOHPGDSCES2CES1HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0000649-B1 5-SUBSTITUTED-1,2-DIHYDRO-3H-PYRROLO(1,2-A)PYRROLE-1-CARBONITRILES AND PROCESS FOR THEIR CONVERSION TO THE CORRESPONDING 1-CARBOXYLIC ACIDS SYNTEX (U.S.A.) INC. (US) 1981-03-25 EP claimed
EP-0000649-B1 5-SUBSTITUTED-1,2-DIHYDRO-3H-PYRROLO(1,2-A)PYRROLE-1-CARBONITRILES AND PROCESS FOR THEIR CONVERSION TO THE CORRESPONDING 1-CARBOXYLIC ACIDS SYNTEX (U.S.A.) INC. (US) 1981-03-25 EP disclosed