SCHEMBL1135151

SCHEMBL1135151

CCCc1ccccc1NC

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADRA2B P18089 1/20 0.45
ADRA2C P18825 1/20 0.45
POLB P06746 3/20 0.41
KDM4E B2RXH2 2/20 0.41
USP2 O75604 1/20 0.41
ALDH1A1 P00352 1/20 0.41
MAPT P10636 1/20 0.41
HPGD P15428 1/20 0.41
RECQL P46063 1/20 0.41
NPSR1 Q6W5P4 1/20 0.41
HSD17B10 Q99714 1/20 0.41
TDP1 Q9NUW8 1/20 0.41
L3MBTL1 Q9Y468 1/20 0.41
AR P10275 1/20 0.40
TAAR1 Q96RJ0 3/20 0.36
ATP4A P20648 1/20 0.36
ATP4B P51164 1/20 0.36
SLC6A2 P23975 1/20 0.36
SLC6A4 P31645 1/20 0.36
SLC6A3 Q01959 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4093561 0.87 CYP3A4 (0.45) ADRA2BADRA2CPOLBKDM4EUSP2
SCHEMBL10407894 0.85 LIPG (0.52) POLB
Hydrochloric Acid SCHEMBL8801544 0.85 CYP3A4 (0.44) ADRA2BADRA2CPOLBKDM4EUSP2
SCHEMBL22535153 0.84 L3MBTL1 (0.43) POLBKDM4EUSP2ALDH1A1MAPT
SCHEMBL13813554 0.84 ADRA2B (0.46) ADRA2BADRA2CKDM4EALDH1A1MAPT
SCHEMBL4093510 0.84 LIPG (0.55)
SCHEMBL4089467 0.84 LIPG (0.55)
SCHEMBL11349035 0.84 LIPG (0.55)
SCHEMBL4083405 0.84 LIPG (0.55)
SCHEMBL4079740 0.84 LIPG (0.55)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 69 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2285769-A1 A PROCESS FOR THE PREPARATION OF ENANTIOMERICALLY PURE AMINES Generics [UK] Limited (GB) 2011-02-23 EP claimed
WO-2009147430-A1 A PROCESS FOR THE PREPARATION OF ENANTIOMERICALLY PURE AMINES GENERICS [UK] LIMITED (GB) 2009-12-10 WO claimed
EP-0344675-A2 Method for the production of selegiline hydrochloride FARMAKON (CS) 1989-12-06 EP claimed
WO-2024124463-A1 PYRROLOPYRIDINE DERIVATIVE, AND PHARMACEUTICAL COMPOSITION THEREOF AND USE THEREOF 武汉睿健医药科技有限公司 2024-06-20 WO disclosed
US-10870657-B2 Compounds for the treatment of cancer and inflammatory disease SHY Therapeutics LLC (US) 2020-12-22 US disclosed
US-20190218229-A1 COMPOUNDS FOR THE TREATMENT OF CANCER AND INFLAMMTORY DISEASE SHY Therapeutics LLC 2019-07-18 US disclosed
US-10239878-B2 Macrocyclic ligands with pendant chelating moieties and complexes thereof LUMIPHORE, INC. (US) 2019-03-26 US disclosed
US-20180194766-A1 MACROCYCLIC LIGANDS WITH PENDANT CHELATING MOIETIES AND COMPLEXES THEREOF LUMIPHORE, INC. 2018-07-12 US disclosed
US-20170260174-A1 Benzene, Pyridine, and Pyridazine Derivatives ESANEX INC (US) 2017-09-14 US disclosed
CN-103732632-B Method for producing olefin block polymer using Group 4 transition metal complex 住友化学株式会社 2017-07-07 CN disclosed
US-9656956-B2 Benzene, pyridine, and pyridazine derivatives ESANEX, INC. (US) 2017-05-23 US disclosed
CN-1537873-A Polyaddition catalyst component, polyaddition catalyst and process for preparing addition polymer ס�ѻ�ѧ��ҵ��ʽ���� 2004-10-20 CN disclosed
CN-1537874-A Polyaddition catalyst component, polyaddition catalyst and method for preparing addition polymer ס�ѻ�ѧ��ҵ��ʽ���� 2004-10-20 CN disclosed
CN-1537872-A Polyaddition catalyst component, polyaddition catalyst, and method for preparing addition polymer ס�ѻ�ѧ��ҵ��ʽ���� 2004-10-20 CN disclosed
CN-1537871-A Polyaddition catalyst component polyaddition catalyst and pruess for producing addition polymer ס�ѻ�ѧ��ҵ��ʽ���� 2004-10-20 CN disclosed
CN-1532209-A Contact product, catalytic component and addition polymerizing cathlyst and method for producing addition polymer 住友化学工业株式会社 2004-09-29 CN disclosed
CN-1530378-A Catalyst component for polyaddition, catalyst and method for producing addition polymer ס�ѻ�ѧ��ҵ��ʽ���� 2004-09-22 CN disclosed
CN-1422286-A Modified particle, support, catalyst component for addition polymerization, catalyst for addition polymerization, and process for producing addition polymer SUMITOMO CHEMICAL CO (JP) 2003-06-04 CN disclosed
CN-1408738-A Catalytic component for addition polymerization, process for producing addition polymerization and process for producing addition polymer SUMITOMO CHEMICAL CO (JP) 2003-04-09 CN disclosed
CN-1306011-A Polyaddition catalyst component, polyaddition catalyst and method for preparing addition polymer SUMITOMO CHEMICAL CO (JP) 2001-08-01 CN disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (5 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20190218229-A1 COMPOUNDS FOR THE TREATMENT OF CANCER AND INFLAMMTORY DISEASE MAPK1, MAPK6, MAP3K1 ADRA2B 3736/4885ADRA2C 3897/4885POLB 1722/4885
US-10870657-B2 Compounds for the treatment of cancer and inflammatory disease MAPK6, MAP3K6, MAPK4 ADRA2B 4143/4885ADRA2C 4307/4885POLB 1589/4885
US-20180194766-A1 MACROCYCLIC LIGANDS WITH PENDANT CHELATING MOIETIES AND COMPLEXES THEREOF TFRC, CLTC, SLC39A3 ADRA2B 4667/4885ADRA2C 4256/4885POLB 1462/4885
US-20170260174-A1 Benzene, Pyridine, and Pyridazine Derivatives CDK4, P2RX4, MKI67 ADRA2B 913/4885ADRA2C 1240/4885POLB 2240/4885
US-10239878-B2 Macrocyclic ligands with pendant chelating moieties and complexes thereof TFRC, CLTC, SLC39A3 ADRA2B 4667/4885ADRA2C 4256/4885POLB 1462/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.