SCHEMBL11399779

SCHEMBL11399779

O=C(O)Cc1nn(-c2ccc(F)cc2)cc1-c1ccc(Br)cc1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RAB9A P51151 3/20 0.44
CCNE1 P24864 1/20 0.43
CDK2 P24941 1/20 0.43
MEN1 O00255 3/20 0.42
KMT2A Q03164 3/20 0.42
NPC1 O15118 2/20 0.42
KDM4E B2RXH2 4/20 0.41
ALDH1A1 P00352 2/20 0.41
HTT P42858 1/20 0.41
SRC P12931 1/20 0.39
BRAF P15056 1/20 0.39
KDR P35968 1/20 0.39
PTGS2 P35354 1/20 0.39
MAPT P10636 2/20 0.38
AGTR1 P30556 1/20 0.38
CA12 O43570 3/20 0.38
CA1 P00915 3/20 0.38
CA2 P00918 3/20 0.38
CA9 Q16790 3/20 0.38
AKR1B1 P15121 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11077918 0.94 RAB9A (0.49) RAB9AMEN1KMT2ANPC1KDM4E
SCHEMBL11764061 0.88 KDM4E (0.50) RAB9ACDK2MEN1KMT2AKDM4E
Pirazolac SCHEMBL153631 0.88 KDM4E (0.51) RAB9ACCNE1CDK2MEN1KMT2A
Pirazolac SCHEMBL10952997 0.86 KDM4E (0.50) RAB9ACCNE1CDK2MEN1KMT2A
SCHEMBL29111861 0.85 RAB9A (0.52) RAB9ACCNE1CDK2MEN1KMT2A
SCHEMBL11764727 0.85 RAB9A (0.64) RAB9ACCNE1CDK2MEN1KMT2A
SCHEMBL11078308 0.83 MEN1 (0.43) RAB9AMEN1KMT2AHTTSRC
SCHEMBL11076213 0.82 PPP1CA (0.49) RAB9AMEN1KMT2AKDM4EALDH1A1
SCHEMBL11443525 0.80 KDM4E (0.56) RAB9AKMT2ANPC1KDM4EALDH1A1
SCHEMBL11764002 0.78 KDM4E (0.60) RAB9AMEN1KMT2AKDM4EALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0022906-A1 Process for the preparation of pyrazole derivatives SCHERING AKTIENGESELLSCHAFT (DE) 1981-01-28 EP claimed