SCHEMBL11432245

SCHEMBL11432245

CN1CCC(=C2c3ccccc3Sc3ccc(Cl)cc32)CC1

nearest known ligand 0.76

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR1A P08908 6/20 0.76
ADRA2A P08913 6/20 0.76
SLC6A2 P23975 6/20 0.76
SLC6A4 P31645 6/20 0.76
ADRA1A P35348 6/20 0.76
DRD3 P35462 6/20 0.76
SLC6A3 Q01959 6/20 0.76
KCNH2 Q12809 6/20 0.76
SETD7 Q8WTS6 5/20 0.76
CHRM2 P08172 5/20 0.76
CHRM1 P11229 5/20 0.76
DRD1 P21728 5/20 0.76
CYP2D6 P10635 5/20 0.76
CYP2C19 P33261 5/20 0.76
OPRM1 P35372 4/20 0.76
TBXA2R P21731 2/20 0.76
ADORA3 P0DMS8 2/20 0.76
CYP3A4 P08684 4/20 0.61
HTT P42858 2/20 0.61
DRD2 P14416 8/20 0.53

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11573081 0.92 SETD7 (0.76) HTR1AADRA2ASLC6A2SLC6A4ADRA1A
Pimethixene SCHEMBL29433731 0.87 SETD7 (1.00) HTR1AADRA2ASLC6A2SLC6A4ADRA1A
Pimethixene SCHEMBL301596 0.87 SETD7 (1.00) HTR1AADRA2ASLC6A2SLC6A4ADRA1A
SCHEMBL11576544 0.86 HTR1A (0.55) HTR1AADRA2ASLC6A2SLC6A4ADRA1A
SCHEMBL11423784 0.85 SETD7 (0.53) HTR1AADRA2ASLC6A2SLC6A4ADRA1A
Hydrochloric Acid SCHEMBL11576537 0.85 HTR1A (0.53) HTR1AADRA2ASLC6A2SLC6A4ADRA1A
SCHEMBL11574868 0.84 DRD3 (0.53) HTR1AADRA2ASLC6A2SLC6A4ADRA1A
SCHEMBL11575971 0.84 SETD7 (0.76) HTR1AADRA2ASLC6A2SLC6A4ADRA1A
SCHEMBL11574284 0.84 SETD7 (0.76) HTR1AADRA2ASLC6A2SLC6A4ADRA1A
SCHEMBL11574597 0.84 LMNA (0.62) HTR1AADRA2ASLC6A2SLC6A4ADRA1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4235916-A ANTIPSYCHOTIC KEFALAS A/S (DK) 1980-11-25 US disclosed
EP-0002902-A1 Methylthiofluorothioxanthene derivative, its preparation and compositions containing it KEFALAS A/S (DK) 1979-07-11 EP disclosed
US-4086350-A FLUORO, CHLORO AND CYANO SUBSTITUTED 4-(9-XANTHENYLIDENE, 9-THIOXANTHENYLIDENE OR 11(6H)-DIBENZO(B,E)OXEPINYLIDENE)-1-METHYL-PIPERIDINES SMITHKLINE CORPORATION (US) 1978-04-25 US disclosed