SCHEMBL11468308

SCHEMBL11468308

CC(C)Oc1nnc(-c2ccc(N(C)C)cc2)c(-c2ccc(N(C)C)cc2)n1

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 1/20 0.37
CYP2C9 P11712 1/20 0.37
CYP2C19 P33261 1/20 0.37
MAPT P10636 6/20 0.37
SMN1; SMN2 Q16637 3/20 0.37
NOX1 Q9Y5S8 1/20 0.36
ALDH1A1 P00352 6/20 0.36
HSD17B10 Q99714 4/20 0.36
KDM4E B2RXH2 4/20 0.36
HPGD P15428 3/20 0.36
ADK P55263 2/20 0.35
KDM5B Q9UGL1 1/20 0.35
LMNA P02545 3/20 0.35
RAB9A P51151 3/20 0.35
GAA P10253 3/20 0.35
MCL1 Q07820 2/20 0.35
NPC1 O15118 2/20 0.35
MAPK1 P28482 1/20 0.35
RECQL P46063 1/20 0.35
TDP1 Q9NUW8 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11478566 0.84 CASR (0.36) MAPTSMN1; SMN2ALDH1A1HSD17B10KDM4E
SCHEMBL11485810 0.82 MAPT (0.45) MAPTSMN1; SMN2NOX1ALDH1A1HSD17B10
SCHEMBL11280072 0.80 NPSR1 (0.47) MAPTSMN1; SMN2ALDH1A1HSD17B10KDM4E
SCHEMBL11468328 0.80 MAPT (0.38) CYP1A2CYP2C9CYP2C19MAPTSMN1; SMN2
SCHEMBL11245322 0.79 ALDH1A1 (0.46) MAPTSMN1; SMN2ALDH1A1KDM4EHPGD
SCHEMBL11244627 0.78 ADK (0.38) CYP1A2CYP2C9CYP2C19MAPTSMN1; SMN2
SCHEMBL11749749 0.76 MAPT (0.40) CYP1A2CYP2C9CYP2C19MAPTALDH1A1
SCHEMBL11485177 0.76 ADK (0.37) CYP1A2CYP2C9CYP2C19NOX1ADK
SCHEMBL11711759 0.76 ALOX5 (0.44) CYP1A2CYP2C9CYP2C19MAPTALDH1A1
SCHEMBL11468266 0.76 MAPT (0.36) CYP1A2MAPTSMN1; SMN2NOX1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4190725-A ANTIINFLAMMATORY ELI LILLY AND COMPANY (US) 1980-02-26 US disclosed
US-4021553-A 5,6-Diaryl-1,2,4-triazines as topically-active anti-inflammatory agents ELI LILLY AND COMPANY (US) 1977-05-03 US disclosed