SCHEMBL1147174

SCHEMBL1147174

COC(=O)CCCCCCN

nearest known ligand 0.64

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
TSHR P16473 3/20 0.64
PAOX Q6QHF9 4/20 0.56
LMNA P02545 4/20 0.55
ALDH1A1 P00352 2/20 0.55
KMT2A Q03164 2/20 0.52
RECQL P46063 2/20 0.52
MEN1 O00255 1/20 0.52
PLG P00747 1/20 0.52
THRB P10828 1/20 0.52
ALOX15 P16050 1/20 0.52
SLC6A2 P23975 1/20 0.52
SLC6A3 Q01959 1/20 0.52
KDM4E B2RXH2 1/20 0.50
CYP1A2 P05177 1/20 0.50
CYP2D6 P10635 1/20 0.48
NFKB1 P19838 1/20 0.48
BLM P54132 1/20 0.46
NPSR1 Q6W5P4 1/20 0.46
L3MBTL1 Q9Y468 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7545025 1.00 TSHR (0.64) TSHRPAOXLMNAALDH1A1KMT2A
SCHEMBL1235539 1.00 TSHR (0.64) TSHRPAOXLMNAALDH1A1KMT2A
SCHEMBL1701715 1.00 TSHR (0.64) TSHRPAOXLMNAALDH1A1KMT2A
SCHEMBL3208419 1.00 TSHR (0.64) TSHRPAOXLMNAALDH1A1KMT2A
SCHEMBL7545108 1.00 TSHR (0.64) TSHRPAOXLMNAALDH1A1KMT2A
SCHEMBL2822938 1.00 TSHR (0.64) TSHRPAOXLMNAALDH1A1KMT2A
SCHEMBL7541388 1.00 TSHR (0.64) TSHRPAOXLMNAALDH1A1KMT2A
SCHEMBL7548607 1.00 TSHR (0.64) TSHRPAOXLMNAALDH1A1KMT2A
SCHEMBL2128896 1.00 TSHR (0.64) TSHRPAOXLMNAALDH1A1KMT2A
SCHEMBL905418 1.00 TSHR (0.64) TSHRPAOXLMNAALDH1A1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 395 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114075187-B Carbonyl pyrazole antitumor compound as well as preparation method and application thereof 山东大学 2023-05-12 CN claimed
CN-115974886-A Macrocyclic lactam compound containing dihydrobenzofuran skeleton and preparation method thereof 国科大杭州高等研究院 2023-04-18 CN claimed
CN-107922352-B Process for preparing protein deacetylase inhibitors 埃斯泰隆制药公司 2021-08-06 CN claimed
EP-3303304-B1 METHODS OF MAKING PROTEIN DEACETYLASE INHIBITORS ACETYLON PHARMACEUTICALS INC (US) 2019-11-20 EP claimed
CN-107619407-B Bis- target spot inhibitor of HDAC and VEGFR based on pazopanib structure and its preparation method and application 山东大学 2019-05-24 CN claimed
US-10144714-B2 Methods of making protein deacetylase inhibitors ACETYLON PHARMACEUTICALS, INC. (US) 2018-12-04 US claimed
EP-3303304-A1 METHODS OF MAKING PROTEIN DEACETYLASE INHIBITORS Acetylon Pharmaceuticals, Inc. (US) 2018-04-11 EP claimed
WO-2016200930-A9 METHODS OF MAKING PROTEIN DEACETYLASE INHIBITORS ACETYLON PHARMACEUTICALS, INC. (US) 2017-02-23 WO claimed
WO-2016200930-A1 METHODS OF MAKING PROTEIN DEACETYLASE INHIBITORS ACETYLON PHARMACEUTICALS, INC. (US) 2016-12-15 WO claimed
US-20160355486-A1 METHODS OF MAKING PROTEIN DEACETYLASE INHIBITORS ACETYLON PHARMACEUTICALS, INC. 2016-12-08 US claimed
US-12479797-B2 Cyclopropyl-amide compounds as dual LSD1/HDAC inhibitors Jubilant Epicore LLC (US) 2025-11-25 US disclosed
EP-3455204-B1 CYCLOPROPYL-AMIDE COMPOUNDS AS DUAL LSD1/HDAC INHIBITORS Jubilant Epicore LLC (US) 2025-10-29 EP disclosed
US-20250302815-A1 PROTEIN TYROSINE PHOSPHATASE TARGETING LIGANDS CALICO LIFE SCIENCES LLC 2025-10-02 US disclosed
CN-119569743-A Compound based on 6-methylfuro [2,3-d ] pyrimidine-4 (3H) -ketone structure, and preparation method and application thereof 沈阳药科大学 2025-03-07 CN disclosed
CN-114380751-B Indanamine derivatives, preparation method and application thereof 上海辉启生物医药科技有限公司 2025-03-07 CN disclosed
US-4244947-A TREATMENT OF ACROMEGALY AND DIABETES AYERST MCKENNA AND HARRISON INC. (CA) 1981-01-13 US disclosed
US-4191754-A ANTIDIABETIC AGENTS, INHIBIT RELEASE OF INSULIN, GLUCAGON AND GROWTH HORMONE MERCK & CO., INC. (US) 1980-03-04 US disclosed
US-4161521-A Somatostatin analogs MERCK & CO., INC. (US) 1979-07-17 US disclosed
US-4102888-A VASODILATORS, ANTITHROMBITIC MERCK & CO., INC. (US) 1978-07-25 US disclosed
US-4059587-A 8-AZA-9-OXO-11-THIA-PROSTANOIC ACID DERIVATIVES; VASODILATORS, ANTICLOTTING, REGULATORS OF IMMUNE RESPONSE MERCK & CO., INC. (US) 1977-11-22 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (4 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-10144714-B2 Methods of making protein deacetylase inhibitors HDAC1, HDAC6, AADAC TSHR 4078/4885PAOX 1153/4885LMNA 2636/4885
US-20250302815-A1 PROTEIN TYROSINE PHOSPHATASE TARGETING LIGANDS PTPN1, PTPN2, PTPN18 TSHR 538/4885PAOX 358/4885LMNA 4758/4885
US-20160355486-A1 METHODS OF MAKING PROTEIN DEACETYLASE INHIBITORS HDAC1, HDAC6, AADAC TSHR 4078/4885PAOX 1153/4885LMNA 2636/4885
US-12479797-B2 Cyclopropyl-amide compounds as dual LSD1/HDAC inhibitors HDAC1, HDAC11, HDAC2 TSHR 2400/4885PAOX 733/4885LMNA 1966/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.