SCHEMBL11477756

SCHEMBL11477756

NC(=S)N(C(=O)c1ccccc1)n1cccn1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.38
TDP1 Q9NUW8 2/20 0.37
L3MBTL1 Q9Y468 2/20 0.37
TSHR P16473 2/20 0.37
POLB P06746 1/20 0.37
CYP3A4 P08684 1/20 0.37
PARP1 P09874 1/20 0.37
MAPT P10636 1/20 0.37
CYP2C19 P33261 1/20 0.37
RECQL P46063 1/20 0.37
BLM P54132 1/20 0.37
PMP22 Q01453 1/20 0.37
HSD17B10 Q99714 1/20 0.37
HTT P42858 1/20 0.35
KMT2A Q03164 3/20 0.34
KDM4E B2RXH2 1/20 0.34
LMNA P02545 1/20 0.34
ADORA3 P0DMS8 1/20 0.34
TMIGD3 P0DMS9 1/20 0.34
CTSL P07711 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27645357 0.71 TDP1 (0.46) ALDH1A1TDP1L3MBTL1TSHRPOLB
SCHEMBL6267389 0.70 TSHR (0.50) ALDH1A1TDP1L3MBTL1TSHRPOLB
SCHEMBL15399512 0.70 PHGDH (0.50) ALDH1A1TSHRMAPTHTTKMT2A
SCHEMBL8723486 0.69 KMT2A (0.53) ALDH1A1TDP1L3MBTL1TSHRPOLB
SCHEMBL11240709 0.69 TSHR (0.48) ALDH1A1TDP1L3MBTL1TSHRPOLB
SCHEMBL2200339 0.68 NPSR1 (0.38) ALDH1A1L3MBTL1TSHRHTTKMT2A
SCHEMBL28761251 0.67 TSHR (0.46) ALDH1A1TDP1L3MBTL1TSHRPOLB
Ethylene SCHEMBL28318847 0.67 TSHR (0.46) ALDH1A1TDP1L3MBTL1TSHRPOLB
SCHEMBL7675958 0.67 SMN1; SMN2 (0.47) ALDH1A1TSHRMAPTHSD17B10HTT
SCHEMBL14120401 0.67 NOS1 (0.33)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4234594-A Pyrazolyl amino imidazolines as antihypertensive agents ABBOTT LABORATORIES (US) 1980-11-18 US disclosed
US-4226773-A Pyrazolyl amino imidazolines as diuretic agents ABBOTT LABORATORIES (US) 1980-10-07 US disclosed
US-4171367-A ANTIINFLAMMATORY ABBOTT LABORATORIES (US) 1979-10-16 US disclosed