SCHEMBL11487530

SCHEMBL11487530

N#Cc1c[nH]nc1[N+](=O)[O-]

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DPP4 P27487 1/20 0.44
VCAM1 P19320 4/20 0.38
MAPT P10636 3/20 0.38
GRIA1 P42261 2/20 0.38
GRIA2 P42262 2/20 0.38
GRIA3 P42263 2/20 0.38
GRIA4 P48058 2/20 0.38
GRM6 O15303 1/20 0.38
CYP1A2 P05177 1/20 0.38
ALOX15 P16050 1/20 0.38
DPYD Q12882 1/20 0.37
POLB P06746 1/20 0.37
CYP2C9 P11712 1/20 0.37
HPGD P15428 1/20 0.37
APEX1 P27695 1/20 0.37
BLM P54132 1/20 0.37
TDP1 Q9NUW8 1/20 0.37
ALDH1A1 P00352 2/20 0.35
HTT P42858 1/20 0.35
XDH P47989 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL43356 0.73 GPR35 (0.38) MAPTGRIA1GRIA2GRIA3GRIA4
SCHEMBL29024294 0.72 VCAM1 (0.43) VCAM1MAPTPOLBHPGDALDH1A1
SCHEMBL3188249 0.71 VCAM1 (0.40) DPP4VCAM1MAPTGRIA1GRIA2
SCHEMBL28116330 0.69
SCHEMBL11561961 0.69
SCHEMBL9324324 0.69
SCHEMBL319993 0.69
SCHEMBL18976164 0.69
SCHEMBL11607215 0.69 MMP2 (0.39) DPP4VCAM1MAPTCYP1A2POLB
Hydrochloric Acid SCHEMBL29060489 0.68 MAPT (0.33) MAPTHTTKMT2AMEN1LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 11 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4145554-A BACTERICIDES, MICROBIOCIDES, HERBICIDES, PARASITICDES ELI LILLY AND COMPANY (US) 1979-03-20 US claimed
CN-108610291-A A kind of preparation method of 3,4- binitropyrazoles 中北大学 2018-10-02 CN disclosed
CN-102250007-A Preparation method of 3,4-binitropyrazole UNIV NORTH CHINA 2011-11-23 CN disclosed
US-4235995-A BACTERIOCIDES, PARASITICIDES, HERBICIDES ELI LILLY AND COMPANY (US) 1980-11-25 US disclosed
US-4235995-A BACTERIOCIDES, PARASITICIDES, HERBICIDES ELI LILLY AND COMPANY (US) 1980-11-25 US disclosed
US-4172136-A FOR URINARY TRACT INFECTIONS BOEHRINGER MANNHEIM GMBH (DE) 1979-10-23 US disclosed
US-4145554-A BACTERICIDES, MICROBIOCIDES, HERBICIDES, PARASITICDES ELI LILLY AND COMPANY (US) 1979-03-20 US disclosed
US-4145554-A BACTERICIDES, MICROBIOCIDES, HERBICIDES, PARASITICDES ELI LILLY AND COMPANY (US) 1979-03-20 US disclosed
US-4105772-A FOR URINARY TRACT INFECTIONS, BACTERICIDES BOEHRINGER MANNHEIM GMBH (DE) 1978-08-08 US disclosed
US-4066776-A Anti-bacterial compositions containing certain 3-nitropyrazoles ELI LILLY AND COMPANY (US) 1978-01-03 US disclosed
US-4066776-A Anti-bacterial compositions containing certain 3-nitropyrazoles ELI LILLY AND COMPANY (US) 1978-01-03 US disclosed