SCHEMBL11489148

SCHEMBL11489148

COc1ccc(CCN(Cc2cc(OC)c(OC)c(OC)c2)C(C)=O)cc1OC

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 3/20 0.55
ALDH1A1 P00352 4/20 0.53
MEN1 O00255 3/20 0.53
KMT2A Q03164 3/20 0.53
MAPT P10636 2/20 0.53
CYP3A4 P08684 2/20 0.52
CYP1A2 P05177 1/20 0.52
CYP2D6 P10635 1/20 0.52
BLM P54132 1/20 0.51
PMP22 Q01453 1/20 0.51
TUBB4A P04350 2/20 0.50
TUBB P07437 2/20 0.50
TUBA3C P0DPH7 2/20 0.50
TUBA1B P68363 2/20 0.50
TUBA4A P68366 2/20 0.50
TUBB4B P68371 2/20 0.50
TUBB3 Q13509 2/20 0.50
TUBB2A Q13885 2/20 0.50
TUBB8 Q3ZCM7 2/20 0.50
TUBA3E Q6PEY2 2/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9542245 0.83 PTGS2 (0.50) MEN1KMT2AGAAAOC3HTR2A
SCHEMBL27590675 0.82 CYP3A4 (0.53) KDM4EALDH1A1MEN1KMT2AMAPT
SCHEMBL16316823 0.78 CYP3A4 (0.52) KDM4EALDH1A1MEN1KMT2AMAPT
SCHEMBL28901341 0.78 L3MBTL1 (0.57) KDM4EALDH1A1MEN1KMT2ASMN1; SMN2
SCHEMBL14276933 0.77 CYP3A4 (0.66) KDM4EALDH1A1MEN1KMT2ACYP3A4
SCHEMBL8233892 0.77 TRPV1 (0.46) KDM4EALDH1A1MEN1KMT2AMAPT
SCHEMBL27591000 0.76 KMT2A (0.49) ALDH1A1MEN1KMT2ACYP3A4CYP1A2
SCHEMBL27590699 0.76 CYP3A4 (0.52) KDM4EALDH1A1MEN1KMT2AMAPT
SCHEMBL8593264 0.75 ALDH1A1 (0.57) ALDH1A1MEN1KMT2AMAPTGAA
SCHEMBL7436339 0.75 TUBB4A (0.76) KDM4EMEN1KMT2ACYP3A4CYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0010119-A1 Isoquinoline derivatives, their preparation and pharmaceutical compositions containing these compounds THE MASSACHUSETTS GENERAL HOSPITAL (US) 1980-04-30 EP disclosed