SCHEMBL114973

SCHEMBL114973

CSc1ccc(CCc2cnc(F)c(B(O)O)c2)cc1

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MMP12 P39900 1/20 0.35
MMP13 P45452 1/20 0.35
CNR2 P34972 1/20 0.33
QPCTL Q9NXS2 1/20 0.33
SMN1; SMN2 Q16637 1/20 0.33
SLC6A4 P31645 4/20 0.33
CGAS Q8N884 1/20 0.32
HTR2A P28223 1/20 0.32
KCNH2 Q12809 1/20 0.32
NPC1 O15118 1/20 0.32
TP53 P04637 1/20 0.32
TSHR P16473 1/20 0.32
RAB9A P51151 1/20 0.32
MAOA P21397 1/20 0.32
SLC6A2 P23975 1/20 0.32
SLC6A3 Q01959 1/20 0.32
ALOX5 P09917 1/20 0.32
GAA P10253 1/20 0.31
MAPT P10636 2/20 0.31
LMNA P02545 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL114587 0.89 SLC6A4 (0.34) SMN1; SMN2SLC6A4NPC1TP53TSHR
SCHEMBL114283 0.73 SLC6A4 (0.39) MMP12MMP13CNR2SLC6A4HTR2A
SCHEMBL114972 0.73 AKR1C3 (0.33) SLC6A4
SCHEMBL12311146 0.73 LPL (0.36) SMN1; SMN2KCNH2NPC1RAB9A
SCHEMBL7817795 0.67 TAAR1 (0.52) SLC6A4MAOASLC6A2SLC6A3
SCHEMBL115669 0.67 SIGMAR1 (0.43) NPC1SLC6A3
SCHEMBL114492 0.67 EGLN1 (0.45) SMN1; SMN2NPC1RAB9AMAPT
SCHEMBL3576871 0.65 AGBL2 (0.35)
SCHEMBL29955213 0.65 AGBL2 (0.35)
SCHEMBL14820681 0.65 CYP1A2 (0.40) TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2424859-A1 INHIBITORS OF PI3 KINASE AND / OR MTOR Amgen, Inc (US) 2012-03-07 EP disclosed
WO-2010126895-A1 INHIBITORS OF PI3 KINASE AND / OR MTOR AMGEN INC. (US) 2010-11-04 WO disclosed