SCHEMBL11516331

SCHEMBL11516331

NC(C(=O)O)c1ccc(Br)cc1Br

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GRM1 Q13255 6/20 0.46
MEN1 O00255 4/20 0.46
KMT2A Q03164 4/20 0.46
TDP1 Q9NUW8 3/20 0.46
CYP1A2 P05177 2/20 0.46
CYP3A4 P08684 1/20 0.43
KDM4E B2RXH2 3/20 0.40
GLA P06280 1/20 0.40
ALOX15 P16050 1/20 0.39
HSD17B10 Q99714 3/20 0.38
CYP2C9 P11712 2/20 0.38
CYP2D6 P10635 1/20 0.38
CYP2C19 P33261 1/20 0.38
GRM8 O00222 1/20 0.38
GRM6 O15303 1/20 0.38
SLC6A2 P23975 1/20 0.38
SLC6A4 P31645 1/20 0.38
DRD3 P35462 1/20 0.38
GRM4 Q14833 1/20 0.38
HSP90AA1 P07900 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28487229 0.79 CRHBP (0.43) GRM1MEN1KMT2ATDP1CYP1A2
SCHEMBL17847415 0.78 DGAT1 (0.44) GRM1MEN1KMT2ATDP1CYP1A2
SCHEMBL25240807 0.76 IDO1 (0.43) GRM1MEN1KMT2ATDP1CYP1A2
SCHEMBL29890267 0.76 IDO1 (0.43) GRM1MEN1KMT2ATDP1CYP1A2
SCHEMBL1439143 0.76 IDO1 (0.43) GRM1MEN1KMT2ATDP1CYP1A2
SCHEMBL30613085 0.73 DGAT1 (0.39) MEN1KMT2ATDP1CYP1A2KDM4E
SCHEMBL28901123 0.71 HSD17B10 (0.52) GRM1MEN1KMT2ATDP1CYP1A2
SCHEMBL8204161 0.71 LMNA (0.42) TDP1ALOX15HSP90AA1TLR9L3MBTL1
SCHEMBL352322 0.71 HSD17B10 (0.52) GRM1MEN1KMT2ATDP1CYP1A2
SCHEMBL352323 0.71 HSD17B10 (0.52) GRM1MEN1KMT2ATDP1CYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4155905-A 6-Substituted penicillanic acid and derivatives thereof E. R. SQUIBB & SONS, INC. (US) 1979-05-22 US disclosed
US-4077967-A 6-Substituted penicillanic acid and derivatives thereof E. R. SQUIBB & SONS, INC. (US) 1978-03-07 US disclosed
US-4061629-A 6-Amino-6-arylthio penicillanic acids and derivatives thereof E. R. SQUIBB & SONS, INC. (US) 1977-12-06 US disclosed
US-4061851-A 7-Amino-7-arylthio cephalosporins E. R. SQUIBB & SONS, INC. (US) 1977-12-06 US disclosed
US-4029669-A 6-Benzalimino-6-arylthio penicillanic acids and derivatives thereof E. R. SQUIBB & SONS, INC. (US) 1977-06-14 US disclosed
US-4026886-A 7-Acyl-7-arylthiocephalosporins E. R. SQUIBB & SONS, INC. (US) 1977-05-31 US disclosed
US-3965093-A 6-Arylthio penicillanic acid and derivatives thereof E. R. SQUIBB & SONS, INC. (US) 1976-06-22 US disclosed
US-3954744-A ANTIBACTERIAL E. R. SQUIBB & SONS, INC. (US) 1976-05-04 US disclosed