SCHEMBL11519925

SCHEMBL11519925

CCc1cnc(NC(=O)NC(=O)c2c(Cl)cccc2Cl)cn1

nearest known ligand 0.46

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
TYK2 P29597 8/20 0.46
JAK2 O60674 7/20 0.46
JAK1 P23458 6/20 0.46
RAB9A P51151 2/20 0.42
NPC1 O15118 1/20 0.42
POLB P06746 1/20 0.40
MAPT P10636 1/20 0.40
GHSR Q92847 1/20 0.40
PPIA P62937 1/20 0.40
HDAC1 Q13547 1/20 0.39
CYP3A4 P08684 1/20 0.39
KDM4E B2RXH2 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11520689 0.87 TYK2 (0.42) TYK2JAK2JAK1RAB9ANPC1
SCHEMBL11524038 0.85 RAB9A (0.41) TYK2JAK2JAK1RAB9ANPC1
SCHEMBL11524573 0.83 RAB9A (0.46) TYK2JAK2JAK1RAB9ANPC1
SCHEMBL11519411 0.83 RAB9A (0.47) TYK2JAK2JAK1RAB9ANPC1
SCHEMBL11521969 0.82 JAK2 (0.42) TYK2JAK2JAK1RAB9ANPC1
SCHEMBL11522976 0.81 RAB9A (0.45) TYK2JAK2JAK1RAB9ANPC1
SCHEMBL11526152 0.80 RAB9A (0.42) TYK2JAK2JAK1RAB9ANPC1
SCHEMBL11163699 0.78 RAB9A (0.68) RAB9ANPC1MAPT
SCHEMBL11523665 0.78 HCRTR1 (0.48) TYK2RAB9ANPC1MAPTKDM4E
SCHEMBL11525363 0.78 CHEK1 (0.54)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4160834-A INSECTICIDES ELI LILLY AND COMPANY (US) 1979-07-10 US disclosed
US-4083977-A Novel insecticidal 1-(substituted benzoyl)-3-(substituted pyrazinyl)ureas ELI LILLY AND COMPANY (US) 1978-04-11 US disclosed