SCHEMBL11532255

SCHEMBL11532255

Cc1ccc(C(=O)c2cc3cc(C(=O)O)oc3c(Cl)c2Cl)s1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.48
DAO P14920 2/20 0.43
PIM1 P11309 1/20 0.36
GPR35 Q9HC97 2/20 0.34
L3MBTL1 Q9Y468 1/20 0.34
ADORA2A P29274 3/20 0.34
ADORA2B P29275 2/20 0.34
POLB P06746 3/20 0.33
KMT2A Q03164 2/20 0.33
RXRA P19793 1/20 0.33
RXRB P28702 1/20 0.33
RXRG P48443 1/20 0.33
TDP1 Q9NUW8 1/20 0.33
TTR P02766 1/20 0.33
MEN1 O00255 1/20 0.33
KDR P35968 2/20 0.32
NPC1 O15118 1/20 0.32
RAB9A P51151 1/20 0.32
SMN1; SMN2 Q16637 1/20 0.32
HPGD P15428 2/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11537169 0.82 PIM1 (0.40) DAOPIM1GPR35POLBTDP1
SCHEMBL11532310 0.79 MAPT (0.48) ALDH1A1DAOGPR35L3MBTL1POLB
SCHEMBL11536698 0.77 ALDH1A1 (0.46) ALDH1A1PIM1POLBKMT2ATDP1
SCHEMBL11532265 0.74 RAB9A (0.50) ALDH1A1PIM1GPR35POLBKMT2A
SCHEMBL11535390 0.73 DAO (0.41) DAOPIM1GPR35POLBHPGD
SCHEMBL11530908 0.73 PIM1 (0.34) DAOPIM1GPR35ADORA2APOLB
SCHEMBL11535276 0.73 NPC1 (0.45) ALDH1A1DAOGPR35L3MBTL1POLB
SCHEMBL10862875 0.69 PIM1 (0.40) ALDH1A1DAOPIM1GPR35POLB
SCHEMBL10852840 0.69 PIM1 (0.37) DAOPIM1GPR35POLBHPGD
SCHEMBL11166639 0.68 PIM1 (0.32) DAOPIM1GPR35POLBHPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4085117-A DIURETIC-SALURETIC, URICOSURIC, HYPOTENSIVE, ANTIKALURETIC AGENTS MERCK & CO., INC. (US) 1978-04-18 US claimed
US-4154742-A DIURETICS MERCK & CO., INC. (US) 1979-05-15 US disclosed
US-4085117-A DIURETIC-SALURETIC, URICOSURIC, HYPOTENSIVE, ANTIKALURETIC AGENTS MERCK & CO., INC. (US) 1978-04-18 US disclosed