SCHEMBL11535925

SCHEMBL11535925

O=C(CC1CSc2ccccc2O1)N1CCC(O)(c2ccccc2)CC1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.42
MEN1 O00255 1/20 0.41
KMT2A Q03164 1/20 0.41
LTA4H P09960 2/20 0.40
OPRL1 P41146 1/20 0.40
HSD11B1 P28845 1/20 0.39
POLB P06746 2/20 0.39
CHRM4 P08173 2/20 0.39
EPHX2 P34913 1/20 0.39
CA12 O43570 1/20 0.38
CA1 P00915 1/20 0.38
CA2 P00918 1/20 0.38
CA7 P43166 1/20 0.38
CA9 Q16790 1/20 0.38
CA14 Q9ULX7 1/20 0.38
SCD5 Q86SK9 1/20 0.38
DRD2 P14416 2/20 0.38
DRD4 P21917 1/20 0.38
DRD3 P35462 1/20 0.38
HPGD P15428 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11537204 0.81 LTA4H (0.52) ALDH1A1LTA4HPOLBDRD2HPGD
SCHEMBL11539863 0.80 OPRL1 (0.47) MEN1KMT2ALTA4HOPRL1POLB
SCHEMBL11638248 0.76 ADRA1A (0.44) ALDH1A1MEN1KMT2APOLBHPGD
SCHEMBL11538594 0.72 HTT (0.58) ALDH1A1LTA4HPOLBDRD2HPGD
SCHEMBL10760411 0.69 OPRM1 (0.66) ALDH1A1MEN1KMT2AOPRL1HSD11B1
SCHEMBL12702280 0.68 MEN1 (0.76) ALDH1A1MEN1KMT2AOPRL1HSD11B1
SCHEMBL11612235 0.67 MEN1 (0.50) ALDH1A1MEN1KMT2AOPRL1HSD11B1
SCHEMBL6097642 0.67 ADRA1A (0.45) MEN1KMT2ADRD3
SCHEMBL9301424 0.67 ADRA1A (0.45) MEN1KMT2AEPHX2
SCHEMBL795975 0.67 ALDH1A1 (0.56) ALDH1A1MEN1KMT2AOPRL1HSD11B1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4140781-A Analgesic and neuraleptic 2-piperidinoalkyl-1,4-benzodioxans CIBA-GEIGY CORPORATION (US) 1979-02-20 US disclosed
US-4129655-A Neuroleptic 2-piperidinoalkyl-1,4-benzodioxans CIBA-GEIGY CORPORATION (US) 1978-12-12 US disclosed
US-4104396-A NEUROLEPTIC, ANALGESIC CIBA-GEIGY CORPORATION (US) 1978-08-01 US disclosed