SCHEMBL9301424

SCHEMBL9301424

O=C(c1ccccc1)N1CCC(CNCC2CSc3ccccc3O2)CC1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADRA1A P35348 3/20 0.45
ADRA1D P25100 2/20 0.45
ADRA1B P35368 2/20 0.45
EPHX1 P07099 2/20 0.44
EPHX2 P34913 2/20 0.44
HDAC3 O15379 1/20 0.44
HDAC4 P56524 1/20 0.44
HDAC1 Q13547 1/20 0.44
HDAC7 Q8WUI4 1/20 0.44
HDAC2 Q92769 1/20 0.44
HDAC10 Q969S8 1/20 0.44
HDAC11 Q96DB2 1/20 0.44
HDAC8 Q9BY41 1/20 0.44
HDAC6 Q9UBN7 1/20 0.44
HDAC9 Q9UKV0 1/20 0.44
HDAC5 Q9UQL6 1/20 0.44
TP53 P04637 1/20 0.43
CYP1A2 P05177 1/20 0.43
CYP3A4 P08684 1/20 0.43
CYP2D6 P10635 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9302190 0.90 MGLL (0.45) ADRA1AADRA1DADRA1BCYP2D6CYP2C19
SCHEMBL9302364 0.89 EPHX2 (0.46) ADRA1AEPHX2TP53CYP1A2CYP3A4
SCHEMBL9301904 0.87 ADRA1A (0.51) ADRA1AADRA1DADRA1BTP53CYP1A2
SCHEMBL9301407 0.81 ADRA1D (0.68) ADRA1AADRA1DADRA1BSMN1; SMN2
SCHEMBL9302494 0.77 ADRA1A (0.49) ADRA1AADRA1DADRA1BTP53CYP1A2
SCHEMBL9301300 0.74 ADRA1D (0.60) ADRA1AADRA1DADRA1B
SCHEMBL9302459 0.73 CXCR4 (0.54) ADRA1AADRA1DADRA1BHDAC8TP53
SCHEMBL9302003 0.73 ADRA1D (0.60) ADRA1AADRA1DADRA1BTSHRSMN1; SMN2
SCHEMBL9301418 0.73 ACHE (0.43) EPHX1EPHX2CYP2C19MEN1KMT2A
SCHEMBL9301885 0.73 CXCR4 (0.56) ADRA1ATP53CYP1A2CYP3A4CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5286735-A Antidepressants, anxiolytic agents PIERRE FABRE MEDICAMENT (FR) 1994-02-15 US claimed
US-5286735-A Antidepressants, anxiolytic agents PIERRE FABRE MEDICAMENT (FR) 1994-02-15 US disclosed