SCHEMBL11545648

SCHEMBL11545648

NC(=O)c1cc2cc3c(cc2nc1N)OCO3

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.54
HPGD P15428 4/20 0.54
KDM4E B2RXH2 4/20 0.54
GLA P06280 1/20 0.54
GAA P10253 1/20 0.54
IKBKB O14920 1/20 0.51
PI4K2A Q9BTU6 1/20 0.43
RAB9A P51151 5/20 0.40
SMN1; SMN2 Q16637 5/20 0.40
MAPT P10636 4/20 0.40
HSD17B10 Q99714 3/20 0.40
KMT2A Q03164 2/20 0.40
TSHR P16473 2/20 0.40
MEN1 O00255 1/20 0.40
TP53 P04637 1/20 0.40
CYP3A4 P08684 1/20 0.40
CYP2D6 P10635 1/20 0.40
CYP2C9 P11712 1/20 0.40
PKM P14618 1/20 0.40
MAPK1 P28482 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6014247 0.79 LMNA (0.53) ALDH1A1HPGDKDM4EGAARAB9A
Urea SCHEMBL6014244 0.76 ALDH1A1 (0.49) ALDH1A1HPGDKDM4ERAB9ASMN1; SMN2
SCHEMBL8223252 0.74 PTPN1 (0.44) ALDH1A1HPGDKDM4EPI4K2ARAB9A
SCHEMBL6014245 0.73 TRPM8 (0.40) ALDH1A1HPGDKDM4EGAAIKBKB
SCHEMBL30682087 0.72 KMT2A (0.46) ALDH1A1HPGDKDM4EGAARAB9A
SCHEMBL7668928 0.71 MAPT (0.50) ALDH1A1HPGDKDM4EGAAPI4K2A
SCHEMBL8352155 0.70 KDM4E (1.00) ALDH1A1HPGDKDM4EGLAGAA
Urea SCHEMBL6014279 0.69 L3MBTL1 (0.42) ALDH1A1HPGDKDM4EGAARAB9A
SCHEMBL8756161 0.69 KDM4E (0.54) ALDH1A1HPGDKDM4EGLAGAA
SCHEMBL30837 0.68 IKBKB (1.00) ALDH1A1HPGDKDM4EGLAGAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4134981-A ANTIALLERGENS PFIZER INC. (US) 1979-01-16 US disclosed
US-4120962-A Fused pyrimidin-4(3H)-ones as antiallergy agents PFIZER INC. (US) 1978-10-17 US disclosed
US-4044134-A FUSED WITH QUINOLINE OR PYRIDINE, 2-METHYL, ETHYL, OR ACETYL GROUP PFIZER INC. (US) 1977-08-23 US disclosed
US-3974161-A Fused pyrimidin-4(3H)-ones as antiallergy agents PFIZER INC. (US) 1976-08-10 US disclosed