SCHEMBL115552

SCHEMBL115552

Nc1cccc2c1C(c1ccccc1)c1ccccc1-2

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.44
L3MBTL1 Q9Y468 1/20 0.44
HSD17B10 Q99714 1/20 0.43
CYP3A4 P08684 3/20 0.41
LMNA P02545 2/20 0.41
CYP1A2 P05177 2/20 0.41
MAPK1 P28482 2/20 0.41
TP53 P04637 1/20 0.41
MAPT P10636 1/20 0.41
HTR2B P41595 1/20 0.41
GID4 Q8IVV7 1/20 0.40
SLC6A2 P23975 3/20 0.37
SLC6A4 P31645 3/20 0.37
SLC6A3 Q01959 3/20 0.37
HTR2A P28223 2/20 0.37
PTGS2 P35354 2/20 0.37
HRH1 P35367 2/20 0.37
RGS12 O14924 1/20 0.37
CYP2D6 P10635 1/20 0.37
ALOX12 P18054 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29377413 1.00 ALDH1A1 (0.44) ALDH1A1L3MBTL1HSD17B10CYP3A4LMNA
SCHEMBL283175 0.81 MAPT (0.38) ALDH1A1L3MBTL1HSD17B10CYP3A4LMNA
SCHEMBL30287378 0.81 CHRNB2 (0.44) ALDH1A1HSD17B10CYP3A4LMNACYP1A2
SCHEMBL150218 0.81 CHRNB2 (0.44) ALDH1A1HSD17B10CYP3A4LMNACYP1A2
SCHEMBL2639173 0.79 MEN1 (0.45) ALDH1A1HSD17B10CYP3A4LMNACYP1A2
SCHEMBL28773419 0.79 HTR2B (0.39) ALDH1A1CYP3A4LMNACYP1A2MAPK1
SCHEMBL6377271 0.79 MAPK1 (0.39) ALDH1A1CYP3A4LMNACYP1A2MAPK1
SCHEMBL28773457 0.79 IDO1 (0.41) ALDH1A1CYP3A4LMNACYP1A2MAPK1
SCHEMBL25171318 0.79 LMNA (0.54) ALDH1A1L3MBTL1HSD17B10CYP3A4LMNA
SCHEMBL70993 0.79 LMNA (0.54) ALDH1A1L3MBTL1HSD17B10CYP3A4LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Appears in 3689 patents — a generic fragment claimed broadly, so it's down-weighted as IP noise. Top by claim status then date:

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-12060334-B2 3-substituted phenazine derivatives as antimicrobial agents UNIVERSITY OF FLORIDA RESEARCH FOUNDATION, INCORPORATED (US) 2024-08-13 US claimed
EP-3715346-B1 THIAZOLYL-CONTAINING COMPOUNDS FOR TREATING PROLIFERATIVE DISEASES DANA FARBER CANCER INST INC (US) 2024-01-03 EP claimed
EP-3606528-B1 TRICYCLIC COMPOUNDS AS GLYCOGEN SYNTHASE KINASE 3 (GSK3) INHIBITORS AND USES THEREOF BROAD INST INC (US) 2023-10-18 EP claimed
EP-3291676-B1 MITRAGYNINE ANALOGS AND USES THEREOF MEMORIAL SLOAN KETTERING CANCER CENTER (US) 2022-08-17 EP claimed
US-11241435-B2 Uses of salt-inducible kinase (SIK) inhibitors for treating osteoporosis THE GENERAL HOSPITAL CORPORATION (US) 2022-02-08 US claimed
EP-3172213-B1 MACROCYCLIC KINASE INHIBITORS AND USES THEREOF DANA FARBER CANCER INST INC (US) 2021-09-22 EP claimed
EP-3092220-B1 VITAMIN C PRODRUGS AND USES THEREOF UNIV FLORIDA (US) 2021-01-20 EP claimed
US-10870651-B2 Inhibitors of cyclin-dependent kinase 7 (CDK7) DANA-FARBER CANCER INSTITUTE, INC. (US) 2020-12-22 US claimed
EP-3171874-B1 IMIDAZOLYL KINASE INHIBITORS AND USES THEREOF DANA FARBER CANCER INST INC (US) 2020-11-18 EP claimed
US-10711036-B2 MALT1 inhibitors and uses thereof CORNELL UNIVERSITY (US) 2020-07-14 US claimed
EP-2550285-B1 TRIOXACARCINS AND USES THEREOF HARVARD COLLEGE (US) 2017-07-19 EP claimed
US-20150376201-A1 CORTISTATIN ANALOGUES AND SYNTHESES THEREOF PRESIDENT AND FELLOWS OF HARVARD COLLEGE (US) 2015-12-31 US claimed
CN-103214409-B The synthesis of tsiklomitsin and analogue thereof PRESIDENT AND FELLOWS OF HARVARD COLLEGE (US) 2015-10-21 CN claimed
EP-1407463-A2 CAPACITOR HAVING EPOXY DIELECTRIC LAYER CURED WITH AMINOPHENYLFLUORENES 3M Innovative Properties Company (US) 2004-04-14 EP claimed
US-6577492-B2 Use of 9,9-bis(aminophenyl)fluorene curing agents reduces water adsorption in the dielectric layer 3M INNOVATIVE PROPERTIES COMPANY 2003-06-10 US claimed
US-20030030966-A1 Capacitor having epoxy dielectric layer cured with aminophenylfluorenes 3M INNOVATIVE PROPERTIES COMPANY 2003-02-13 US claimed
WO-2003007319-A2 CAPACITOR HAVING EPOXY DIELECTRIC LAYER CURED WITH AMINOPHENYLFLUORENES 3M INNOVATIVE PROPERTIES COMPANY (US) 2003-01-23 WO claimed
EP-0203828-B1 EPOXY RESIN CURING AGENT, CURING PROCESS AND COMPOSITION CONTAINING IT MINNESOTA MINING AND MANUFACTURING COMPANY (US) 1990-03-28 EP claimed
US-4684678-A POLYEPOXIDES OF HIGH GLASS TRANSITION TEMPERATURE AND DUCTILITY MINNESOTA MINING AND MANUFACTURING COMPANY (US) 1987-08-04 US claimed
EP-0203828-A1 Epoxy resin curing agent, curing process and composition containing it MINNESOTA MINING AND MANUFACTURING COMPANY (US) 1986-12-03 EP claimed