SCHEMBL11563201

SCHEMBL11563201

[O]c1ccc2c(-c3cccc(F)c3F)noc2c1Cl

nearest known ligand 0.38

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
PTGS1 P23219 1/20 0.38
BCAT1 P54687 1/20 0.36
CYP17A1 P05093 4/20 0.33
GABRA5 P31644 1/20 0.32
MAPT P10636 1/20 0.32
GPBAR1 Q8TDU6 2/20 0.31
ESR1 P03372 3/20 0.31
ESR2 Q92731 3/20 0.31
PDE3B Q13370 1/20 0.30
PDE3A Q14432 1/20 0.30
APEX1 P27695 1/20 0.30
CCNE2 O96020 1/20 0.30
CCNE1 P24864 1/20 0.30
CDK2 P24941 1/20 0.30
HTR7 P34969 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11558673 0.89 PTGS1 (0.45) PTGS1CYP17A1GABRA5MAPTGPBAR1
SCHEMBL11560465 0.86 PTGS1 (0.36) PTGS1MAPTGPBAR1
SCHEMBL11557773 0.83 BCAT1 (0.36) PTGS1BCAT1CYP17A1GABRA5ESR1
SCHEMBL10664082 0.83 ESR1 (0.36) PTGS1BCAT1CYP17A1ESR1ESR2
SCHEMBL10655633 0.80 HTR3A (0.39) PTGS1BCAT1CYP17A1
SCHEMBL11557764 0.80 ESR1 (0.40) CYP17A1MAPTESR1ESR2
SCHEMBL11560451 0.80 HSD17B10 (0.43) PTGS1CYP17A1MAPTGPBAR1HTR7
SCHEMBL11558263 0.78 GABRA5 (0.35) PTGS1GABRA5GPBAR1APEX1
SCHEMBL11560540 0.78 PTGS1 (0.33) PTGS1CYP17A1GABRA5PDE3BPDE3A
SCHEMBL11558638 0.78 MAPK14 (0.37) GABRA5MAPTPDE3BPDE3A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0002666-A1 1,2-Benzisoxazolyloxy (or thio) acetic acids and related compounds, process for their preparation and medicines containing them HOECHST AKTIENGESELLSCHAFT (DE) 1979-07-11 EP disclosed