SCHEMBL11565945

SCHEMBL11565945

CC1=C(OC(=O)O)C(c2cccs2)C(OC(=O)O)=C(C)N1

nearest known ligand 0.57

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 7/20 0.51
MAPT P10636 2/20 0.51
KMT2A Q03164 2/20 0.51
MEN1 O00255 1/20 0.51
L3MBTL1 Q9Y468 1/20 0.45
KDM4E B2RXH2 4/20 0.43
HSD17B10 Q99714 3/20 0.43
PKM P14618 1/20 0.42
HPGD P15428 2/20 0.42
GAA P10253 2/20 0.42
ADORA2B P29275 5/20 0.41
TSHR P16473 2/20 0.41
LMNA P02545 1/20 0.41
POLB P06746 1/20 0.41
AGTR1 P30556 1/20 0.41
ADORA3 P0DMS8 1/20 0.40
NR3C1 P04150 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9690862 0.85 ALDH1A1 (0.54) ALDH1A1MAPTKMT2AMEN1L3MBTL1
SCHEMBL10863780 0.76 TP53 (0.38) ALDH1A1MAPTKMT2AMEN1KDM4E
SCHEMBL7815170 0.75 ALDH1A1 (0.59) ALDH1A1MAPTKMT2AMEN1L3MBTL1
SCHEMBL7273862 0.73 ALDH1A1 (0.60) ALDH1A1MAPTKMT2AMEN1L3MBTL1
SCHEMBL1666306 0.72 ALDH1A1 (0.74) ALDH1A1MAPTKMT2AMEN1L3MBTL1
SCHEMBL11500155 0.72 ALDH1A1 (0.44) ALDH1A1MAPTKMT2AMEN1L3MBTL1
SCHEMBL7818024 0.70 ALDH1A1 (0.62) ALDH1A1MAPTKMT2AMEN1HSD17B10
SCHEMBL9691613 0.70 ADORA3 (0.49) ALDH1A1MAPTKMT2AMEN1KDM4E
SCHEMBL7266747 0.70 KDM4E (0.56) ALDH1A1MAPTKMT2AMEN1L3MBTL1
SCHEMBL7267057 0.69 L3MBTL1 (0.65) ALDH1A1MAPTKMT2AMEN1L3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0001769-A1 Sulfur-containing esters of 1,4-dihydropyridine carboxylic acids, their preparation and pharmaceutical use BAYER AG (DE) 1979-05-16 EP disclosed