SCHEMBL11577388

SCHEMBL11577388

C#CCN1CCN(C2Cc3ccc(OC)cc3Oc3ccc(C)cc32)CC1

nearest known ligand 0.38

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
MAOB P27338 2/20 0.38
HRH3 Q9Y5N1 1/20 0.37
MTNR1B P49286 3/20 0.36
ALDH1A1 P00352 1/20 0.35
MTNR1A P48039 2/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL11577946 0.99 MAOB (0.37) MAOBHRH3MTNR1BALDH1A1MTNR1A
SCHEMBL11576248 0.85 HRH3 (0.42) HRH3MTNR1B
SCHEMBL11575657 0.82 ALDH1A1 (0.47) MTNR1BALDH1A1MTNR1A
SCHEMBL11575922 0.81 HTR3A (0.41)
SCHEMBL11576273 0.79 NQO2 (0.40) HRH3ALDH1A1
SCHEMBL11576126 0.78 NQO2 (0.39) HRH3ALDH1A1
SCHEMBL11577392 0.73 POLB (0.43) MAOBHRH3
SCHEMBL11599293 0.71 POLB (0.49) MTNR1BALDH1A1MTNR1A
SCHEMBL11682864 0.70 DRD2 (0.41) ALDH1A1
SCHEMBL11794419 0.70 DRD2 (0.52) ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4032525-A CNS DEPRESSANTS, NEUROLEPTICS HOFFMANN-LA ROCHE INC. (US) 1977-06-28 US claimed
US-4118572-A CNS DEPRESSANTS, NEUROLEPTIC AGENTS, SCHIZOPHRENIA, TRANQUILIZERS HOFFMANN-LA ROCHE INC. (US) 1978-10-03 US disclosed
US-4105664-A Dibenz[b,f]oxepin derivatives HOFFMANN-LA ROCHE INC. (US) 1978-08-08 US disclosed
US-4100173-A DEPRESSANTS, SCHIZOPHRENIA, TRANQUILIZERS HOFFMANN-LA ROCHE INC. (US) 1978-07-11 US disclosed
US-4091023-A ANTISCHIZOPHRENIA AGENTS, TRANQUILIZERS HOFFMANN-LA ROCHE INC. (US) 1978-05-23 US disclosed