SCHEMBL11580765

SCHEMBL11580765

N=C(NC(N)=O)Nc1c(Cl)cc(I)cc1Cl

nearest known ligand 0.36

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 2/20 0.36
PLAU P00749 1/20 0.33
NPC1 O15118 1/20 0.31
ADRA2A P08913 1/20 0.30
CYP2D6 P10635 1/20 0.30
ADRA2B P18089 1/20 0.30
ADRA2C P18825 1/20 0.30
HTR1D P28221 1/20 0.30
HTR1B P28222 1/20 0.30
NISCH Q9Y2I1 1/20 0.30
BCAT2 O15382 1/20 0.30
PLK1 P53350 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11579559 0.90 CYP1A2 (0.32) CYP1A2PLAUNPC1
SCHEMBL11091737 0.86 ALDH1A1 (0.40) CYP1A2PLAUNPC1
SCHEMBL11579652 0.83 CYP1A2 (0.36) CYP1A2NPC1BCAT2PLK1
SCHEMBL11086646 0.83 HTT (0.44) CYP1A2PLAU
SCHEMBL11097728 0.83 CYP1A2 (0.36) CYP1A2PLAUNPC1
SCHEMBL11583012 0.83 RAB9A (0.35) CYP1A2PLAUNPC1
SCHEMBL11420556 0.80 CYP1A2 (0.36) CYP1A2PLAUNPC1ADRA2ACYP2D6
SCHEMBL11580439 0.80 CYP1A2 (0.43) CYP1A2NPC1
Biclodil SCHEMBL1815631 0.79 CYP1A2 (0.49) CYP1A2PLAU
SCHEMBL11091069 0.78 ALDH1A1 (0.45) CYP1A2PLAUNPC1ADRA2ACYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4088785-A HYPOTENSIVE AGENTS WILLIAM H. RORER, INC. (US) 1978-05-09 US disclosed