SCHEMBL11601474

SCHEMBL11601474

COc1ccc2nc(OC(C)C)n[n+]([O-])c2c1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CRHBP P24387 1/20 0.50
CRHR2 Q13324 1/20 0.50
KEAP1 Q14145 1/20 0.50
NFE2L2 Q16236 1/20 0.50
CYP2C19 P33261 8/20 0.39
CYP2E1 P05181 7/20 0.39
CYP2C8 P10632 7/20 0.39
CYP2D6 P10635 7/20 0.39
CYP2C9 P11712 7/20 0.39
CYP2B6 P20813 7/20 0.39
CYP1A2 P05177 7/20 0.39
CYP3A4 P08684 7/20 0.39
KDM4E B2RXH2 3/20 0.38
ALDH1A1 P00352 2/20 0.38
POLB P06746 2/20 0.38
SMN1; SMN2 Q16637 2/20 0.38
KMT2A Q03164 2/20 0.38
NQO2 P16083 2/20 0.38
MEN1 O00255 1/20 0.38
NPC1 O15118 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11603037 0.89 CRHBP (0.43) CRHBPCRHR2KEAP1NFE2L2CYP2C19
SCHEMBL11603107 0.81 GABRP (0.37) CYP1A2CYP3A4KDM4EALDH1A1POLB
SCHEMBL11601677 0.81 LMNA (0.35) CRHBPCRHR2KEAP1NFE2L2ALDH1A1
SCHEMBL6674577 0.78 CRHBP (0.54) CRHBPCRHR2KEAP1NFE2L2CYP2C19
SCHEMBL10612622 0.78 CRHBP (0.54) CRHBPCRHR2KEAP1NFE2L2CYP2C19
SCHEMBL11331634 0.73 CRHBP (0.49) CRHBPCRHR2KEAP1NFE2L2KDM4E
SCHEMBL11602714 0.70 MAT2A (0.46) CRHBPCRHR2KEAP1NFE2L2CYP2C19
SCHEMBL29216871 0.68 CRHBP (0.45) CRHBPCRHR2KEAP1NFE2L2KDM4E
SCHEMBL6833397 0.68 CRHBP (0.43) CRHBPCRHR2KEAP1NFE2L2POLB
SCHEMBL15010394 0.67 CRHBP (1.00) CRHBPCRHR2KEAP1NFE2L2CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4067981-A FUNGICIDES, BACTERICIDES, INSECTICIDES, ACARICIDES BAYER AKTIENGESELLSCHAFT (DT) 1978-01-10 US disclosed