SCHEMBL11625367

SCHEMBL11625367

CS(=O)(=O)Nc1ccc(-c2nc(C(F)(F)F)c[nH]2)cc1

nearest known ligand 0.54

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
KIF11 P52732 6/20 0.54
PTGS2 P35354 7/20 0.47
ALOX5 P09917 1/20 0.44
MAP2K4 P45985 1/20 0.42
HPGD P15428 1/20 0.42
IKBKB O14920 2/20 0.41
CHUK O15111 2/20 0.41
CLK1 P49759 1/20 0.41
DYRK1A Q13627 1/20 0.41
DYRK2 Q92630 1/20 0.41
DYRK1B Q9Y463 1/20 0.41
PIP4K2A P48426 1/20 0.41
PIP4K2B P78356 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6532907 0.82 PTGS2 (0.50) KIF11PTGS2
SCHEMBL11623789 0.80 HPGD (0.43) HPGD
SCHEMBL11123090 0.77 KIF11 (0.51) KIF11PTGS2
SCHEMBL27731893 0.76 NPBWR1 (0.44) PTGS2HPGD
SCHEMBL26093883 0.74 KDM4E (0.44) HPGD
SCHEMBL8797359 0.74 GFER (0.50) KIF11HPGD
SCHEMBL25250074 0.72 KIF11 (0.43) KIF11HPGD
SCHEMBL11626212 0.72 KIF11 (0.42) KIF11HPGD
SCHEMBL3095172 0.72 HPGD (0.38) PTGS2HPGD
SCHEMBL27731900 0.72 KDM4E (0.45) PTGS2HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4125530-A FROM 1,1-DIHALO-3,3,3-TRIFLUOROACETONE, BASE, AMMONIA AND A CARBOXALDEHYDE MERCK & CO., INC. (US) 1978-11-14 US disclosed
US-4032522-A ANTI-GOUT, ANTI-HYPERURICEMIC MERCK & CO., INC. (US) 1977-06-28 US disclosed