SCHEMBL11630143

SCHEMBL11630143

O=CNc1ccc(Cl)cc1C(=O)c1ccccc1Cl

nearest known ligand 0.61

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GABRP O00591 2/20 0.61
GABRD O14764 2/20 0.61
GABRA1 P14867 2/20 0.61
GABRB1 P18505 2/20 0.61
GABRG2 P18507 2/20 0.61
GABRB3 P28472 2/20 0.61
GABRA5 P31644 2/20 0.61
GABRA3 P34903 2/20 0.61
GABRA2 P47869 2/20 0.61
GABRB2 P47870 2/20 0.61
GABRA4 P48169 2/20 0.61
GABRE P78334 2/20 0.61
GABRA6 Q16445 2/20 0.61
GABRG1 Q8N1C3 2/20 0.61
GABRG3 Q99928 2/20 0.61
GABRQ Q9UN88 2/20 0.61
RECQL P46063 1/20 0.59
MAPT P10636 5/20 0.57
CYP1A2 P05177 1/20 0.56
CYP2C19 P33261 1/20 0.56

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11457524 0.84 MAPT (0.62) MAPTCYP1A2CYP2C19ALDH1A1LMNA
SCHEMBL9726995 0.82 GABRP (0.64) GABRPGABRDGABRA1GABRB1GABRG2
SCHEMBL11824528 0.81 GABRP (0.71) GABRPGABRDGABRA1GABRB1GABRG2
SCHEMBL12165506 0.80 TSHR (0.52) MAPTCYP1A2CYP2C19ALDH1A1LMNA
SCHEMBL12165535 0.79 IRAK4 (0.45) GABRPGABRDGABRA1GABRB1GABRG2
SCHEMBL11842389 0.79 RECQL (0.77) GABRPGABRDGABRA1GABRB1GABRG2
SCHEMBL11866382 0.78 MAPT (0.55) RECQLMAPTCYP1A2CYP2C19ALDH1A1
SCHEMBL9851141 0.77 RECQL (0.74) GABRPGABRDGABRA1GABRB1GABRG2
SCHEMBL2991610 0.77 GABRP (0.78) GABRPGABRDGABRA1GABRB1GABRG2
SCHEMBL11061295 0.76 GABRP (1.00) GABRPGABRDGABRA1GABRB1GABRG2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4082764-A Methods for the production of 4H-s-triazolo[4,3-a][1,4]benzodiazepine 5N-oxides TAKEDA CHEMICAL INDUSTRIES, LTD. (JA) 1978-04-04 US disclosed