SCHEMBL11716633

SCHEMBL11716633

COc1ccc2c(c1OC)CCC(NC(C)=O)C2O

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MTNR1A P48039 7/20 0.46
MTNR1B P49286 7/20 0.46
LMNA P02545 3/20 0.45
KDM4E B2RXH2 1/20 0.45
POLB P06746 1/20 0.45
MAPT P10636 1/20 0.45
PARP1 P09874 1/20 0.42
NQO2 P16083 1/20 0.40
CYP2C9 P11712 2/20 0.40
TSHR P16473 2/20 0.40
TUBB1 Q9H4B7 2/20 0.40
MITF O75030 1/20 0.40
KMT2A Q03164 1/20 0.40
GMNN O75496 1/20 0.40
SLC22A3 O75751 1/20 0.40
TUBB4A P04350 1/20 0.40
TP53 P04637 1/20 0.40
CYP1A2 P05177 1/20 0.40
TUBB P07437 1/20 0.40
CYP3A4 P08684 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2465015 0.83 LMNA (0.57) MTNR1AMTNR1BLMNAKDM4EPOLB
SCHEMBL8501371 0.83 LMNA (0.57) MTNR1AMTNR1BLMNAKDM4EPOLB
SCHEMBL8502533 0.83 LMNA (0.57) MTNR1AMTNR1BLMNAKDM4EPOLB
SCHEMBL11721603 0.81 DRD2 (0.46) MTNR1AMTNR1BLMNAKDM4EPARP1
SCHEMBL11717346 0.78 ADRB2 (0.37) MTNR1AMTNR1BLMNAKDM4EPOLB
SCHEMBL24733606 0.76 MTNR1A (0.40) MTNR1AMTNR1BLMNAKDM4EPOLB
SCHEMBL11594202 0.76 DRD2 (0.52) KDM4EKMT2ACYP1A2CYP2D6
SCHEMBL11594200 0.76 DRD2 (0.52) KDM4EKMT2ACYP1A2CYP2D6
SCHEMBL11594197 0.76 DRD2 (0.52) KDM4EKMT2ACYP1A2CYP2D6
SCHEMBL10205808 0.75 PARP1 (0.47) MTNR1AMTNR1BLMNAKDM4EPOLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4041079-A Bicyclic compounds TAKEDA CHEMICAL INDUSTRIES, LTD. (JA) 1977-08-09 US disclosed