SCHEMBL11717643

SCHEMBL11717643

CCC12c3ccccc3C(CC)(c3cc(C(F)(F)F)ccc31)N2C

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KIF11 P52732 1/20 0.40
PDE2A O00408 1/20 0.36
DRD2 P14416 4/20 0.34
KDM4E B2RXH2 1/20 0.34
ALDH1A1 P00352 1/20 0.34
KDM1A O60341 1/20 0.34
RCOR1 Q9UKL0 1/20 0.34
HTR7 P34969 1/20 0.34
CCR6 P51684 1/20 0.33
NPC1 O15118 1/20 0.33
ABCB11 O95342 1/20 0.33
TP53 P04637 1/20 0.33
CYP1A2 P05177 1/20 0.33
CHRM2 P08172 1/20 0.33
ABCB1 P08183 1/20 0.33
HTR1A P08908 1/20 0.33
ADRA2A P08913 1/20 0.33
ADORA3 P0DMS8 1/20 0.33
CYP2D6 P10635 1/20 0.33
CHRM1 P11229 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11720987 0.79 PARK7 (0.37) KDM4EHTR7CYP1A2MAPK1RAB9A
SCHEMBL11715464 0.77 PDK2 (0.36) ALDH1A1TSHRSIGMAR1
SCHEMBL11715541 0.76 MEN1 (0.39) KDM4EALDH1A1HTR7HTR1AADRA2A
SCHEMBL11719254 0.76 PGR (0.38) HTR7
SCHEMBL11721089 0.76 GABRA1 (0.33) SIGMAR1
SCHEMBL11714685 0.76 MEN1 (0.36) ALDH1A1TP53SIGMAR1
SCHEMBL11715899 0.71 PGR (0.31) KDM1ASIGMAR1
SCHEMBL11718223 0.70 MAPT (0.46) ALDH1A1CYP1A2CYP2D6TSHR
SCHEMBL11717928 0.69 ACHE (0.34) NPC1RAB9A
SCHEMBL11714996 0.69 HTR2A (0.33) KDM4ECYP1A2CYP2D6MAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4064139-A TRANQUILIZERS, ANTICONVULSANTS, MUSCLE RELAXANTS, ANTI-PARKINSON'S DISEASE MERCK & CO., INC. (US) 1977-12-20 US claimed
US-4064139-A TRANQUILIZERS, ANTICONVULSANTS, MUSCLE RELAXANTS, ANTI-PARKINSON'S DISEASE MERCK & CO., INC. (US) 1977-12-20 US disclosed