SCHEMBL11735657

SCHEMBL11735657

Nc1ccc2c(c1)C(=O)C[C@H]1CCNC[C@@H]1C2

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CASP1 P29466 1/20 0.34
CASP7 P55210 1/20 0.34
HSD17B10 Q99714 1/20 0.34
CRBN Q96SW2 2/20 0.34
HTR2A P28223 7/20 0.33
HTR2C P28335 6/20 0.33
HTR2B P41595 5/20 0.33
PSEN1 P49768 1/20 0.32
PSEN2 P49810 1/20 0.32
APH1B Q8WW43 1/20 0.32
NCSTN Q92542 1/20 0.32
APH1A Q96BI3 1/20 0.32
PSENEN Q9NZ42 1/20 0.32
PARP1 P09874 1/20 0.32
CA9 Q16790 1/20 0.32
TYMS P04818 1/20 0.32
PRKCZ Q05513 1/20 0.31
DDB1 Q16531 1/20 0.31
MEN1 O00255 1/20 0.31
MAPT P10636 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11735670 1.00 CASP1 (0.34) CASP1CASP7HSD17B10CRBNHTR2A
SCHEMBL11740282 0.73 DRD1 (0.42) HTR2ACA9MAPTKMT2AHTR1A
SCHEMBL11740277 0.73 DRD1 (0.42) HTR2ACA9MAPTKMT2AHTR1A
SCHEMBL448237 0.71 CHRNB2 (0.39) HTR2AHTR2CPSEN1PSEN2APH1B
SCHEMBL3886540 0.68 ADRA2A (0.39) HTR2AHTR2CHTR2B
SCHEMBL27723083 0.67 HTR2C (0.43) HTR2AHTR2CHTR2B
SCHEMBL11732725 0.67
SCHEMBL11732714 0.67
SCHEMBL11533307 0.65 ACHE (0.50) HTR2AHTR2CHTR2BDRD2
SCHEMBL11533311 0.65 ACHE (0.50) HTR2AHTR2CHTR2BDRD2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4034095-A ANTIDEPRESSANT, ANTICHOLINERGIC SANDOZ LTD. (CH) 1977-07-05 US claimed