SCHEMBL11737870

SCHEMBL11737870

COc1c(C)ccc2[nH]c(C(=O)O)cc12

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 5/20 0.49
ALDH1A1 P00352 5/20 0.49
HPGD P15428 4/20 0.49
LMNA P02545 3/20 0.49
HSD17B10 Q99714 2/20 0.49
PIN1 Q13526 1/20 0.47
NGFR P08138 1/20 0.44
FLT3 P36888 1/20 0.44
MEN1 O00255 3/20 0.44
KMT2A Q03164 3/20 0.44
GAA P10253 2/20 0.44
GRIN2D O15399 1/20 0.44
GRIN3B O60391 1/20 0.44
CYP1A2 P05177 1/20 0.44
GLA P06280 1/20 0.44
MAPK1 P28482 1/20 0.44
CYP2C19 P33261 1/20 0.44
AHR P35869 1/20 0.44
CHRNA7 P36544 1/20 0.44
GRIN1 Q05586 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16030401 0.86 CYP1A2 (0.45) KDM4EALDH1A1HPGDLMNAHSD17B10
SCHEMBL16031847 0.86 FLT3 (0.43) KDM4EALDH1A1HPGDLMNAFLT3
SCHEMBL6240318 0.84 KDM4E (0.60) KDM4EALDH1A1HPGDLMNAHSD17B10
SCHEMBL30403281 0.84 KDM4E (0.60) KDM4EALDH1A1HPGDLMNAHSD17B10
SCHEMBL11742020 0.83 PLA2G4A (0.44) KDM4EALDH1A1HPGDLMNAHSD17B10
SCHEMBL2492396 0.83 IDO1 (0.51) KDM4EALDH1A1HPGDLMNAHSD17B10
SCHEMBL11743428 0.83 RHEB (0.51) KDM4EALDH1A1HPGDLMNAHSD17B10
SCHEMBL3107966 0.80 ALDH1A1 (0.54) KDM4EALDH1A1HPGDLMNAHSD17B10
SCHEMBL8913109 0.79 SRD5A2 (0.63) KDM4EALDH1A1HPGDLMNAHSD17B10
SCHEMBL8911576 0.79 KDM4E (0.53) KDM4EALDH1A1HPGDLMNAHSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4060626-A Indole-carboxylic carbon compounds and pharmaceutical compositions containing them BOEHRINGER MANNHEIM G.M.B.H. (DT) 1977-11-29 US claimed
US-4060626-A Indole-carboxylic carbon compounds and pharmaceutical compositions containing them BOEHRINGER MANNHEIM G.M.B.H. (DT) 1977-11-29 US disclosed